SCHEMBL4242154

SCHEMBL4242154

CC(C)NS(=O)(=O)CCN

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.36
SLC6A6 P31641 1/20 0.36
CYP2C19 P33261 1/20 0.36
BLM P54132 1/20 0.36
TRPA1 O75762 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21236263 0.86 APP (0.41) LMNAALDH1A1
SCHEMBL26144799 0.80
SCHEMBL20942663 0.78 CA1 (0.30)
SCHEMBL805360 0.77 ACACB (0.37) CYP2C19
SCHEMBL12138293 0.75 MEN1 (0.33) ALDH1A1
SCHEMBL20942728 0.75 NLRP3 (0.32)
SCHEMBL25932730 0.75 PTGS1 (0.36)
SCHEMBL20034868 0.75 CA2 (0.30)
SCHEMBL10106473 0.73 HPGD (0.38) LMNAALDH1A1HPGD
SCHEMBL15672832 0.73 GRIA1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11591301-B2 Indoleamine-2,3-dioxygenase inhibitor, preparation method therefor and use thereof HINOVA PHARMACEUTICALS INC. (CN) 2023-02-28 US disclosed
US-11180504-B2 Substituted carbapenems for the treatment of bacterial infections ORCHID PHARMA LTD. (IN) 2021-11-23 US disclosed
US-20210047281-A1 INDOLEAMINE-2,3-DIOXYGENASE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF HINOVA PHARMACEUTICALS INC. (CN) 2021-02-18 US disclosed
WO-2019149255-A1 INDOLEAMINE-2,3-DIOXYGENASE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 成都海创药业有限公司 2019-08-08 WO disclosed
US-20090209522-A1 Heterocyclic Non-Peptide GNRH Antagonists TAKEDA CAMBRIDGE LIMITED (GB) 2009-08-20 US disclosed
US-20090209522-A1 Heterocyclic Non-Peptide GNRH Antagonists TAKEDA CAMBRIDGE LIMITED (GB) 2009-08-20 US disclosed
US-20090209522-A1 Heterocyclic Non-Peptide GNRH Antagonists TAKEDA CAMBRIDGE LIMITED (GB) 2009-08-20 US disclosed
EP-1896465-A1 HETEROCYCLIC NON-PEPTIDE GNRH ANTAGONISTS Takeda Cambridge Limited (GB) 2008-03-12 EP disclosed
WO-2007000582-A1 HETEROCYCLIC NON-PEPTIDE GNRH ANTAGONISTS TAKEDA CAMBRIDGE LIMITED (GB) 2007-01-04 WO disclosed
WO-2007000582-A1 HETEROCYCLIC NON-PEPTIDE GNRH ANTAGONISTS TAKEDA CAMBRIDGE LIMITED (GB) 2007-01-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11180504-B2 Substituted carbapenems for the treatment of bacterial infections SLC11A2, GSK3B, GSK3A LMNA 564/4885SLC6A6 3774/4885CYP2C19 113/4885
US-11591301-B2 Indoleamine-2,3-dioxygenase inhibitor, preparation method therefor and use thereof IDO1, IDO2, TPH1 LMNA 3797/4885SLC6A6 2990/4885CYP2C19 52/4885
US-20210047281-A1 INDOLEAMINE-2,3-DIOXYGENASE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF IDO1, IDO2, TPH1 LMNA 3797/4885SLC6A6 2990/4885CYP2C19 52/4885
US-20090209522-A1 Heterocyclic Non-Peptide GNRH Antagonists GNRHR, GHRHR, FSHR LMNA 2647/4885SLC6A6 4864/4885CYP2C19 1924/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.