SCHEMBL4244486

SCHEMBL4244486

COC(=O)c1ccc(OC(=O)C(N)c2ccccc2-c2ccccc2C(=O)O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.47
ALDH1A1 P00352 2/20 0.47
POLB P06746 2/20 0.43
MAPT P10636 3/20 0.42
RAB9A P51151 2/20 0.42
SLC6A3 Q01959 1/20 0.42
KDM4E B2RXH2 2/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
ATM Q13315 1/20 0.41
TSHR P16473 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.41
MEN1 O00255 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
ELANE P08246 2/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
PRTN3 P24158 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4237016 0.86 MYC (0.41) KMT2AALDH1A1MAPTRAB9AKDM4E
SCHEMBL4242290 0.82 MAPK1 (0.48) KMT2AALDH1A1RAB9AKDM4EGAA
SCHEMBL498660 0.74 MYC (0.42) ALDH1A1MAPTKDM4EGAAHPGD
SCHEMBL4239362 0.73 PTPN11 (0.52) KMT2AALDH1A1POLBKDM4ETSHR
SCHEMBL6713222 0.72 SLC6A3 (0.59) KMT2AALDH1A1MAPTRAB9ASLC6A3
SCHEMBL4244489 0.72 KCNA5 (0.57) KMT2AALDH1A1POLBMAPTRAB9A
Phthalic Acid SCHEMBL3454567 0.72 TSHR (0.72) KMT2AALDH1A1POLBMAPTRAB9A
SCHEMBL4241475 0.71 MYC (0.44) KMT2AALDH1A1MAPTGAASMN1; SMN2
SCHEMBL2207409 0.71 ALDH1A1 (0.51) KMT2AALDH1A1MAPTRAB9ASLC6A3
SCHEMBL9480620 0.70 KMT2A (0.79) KMT2AALDH1A1POLBMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090192096-A1 2'-Substituted 1,1'-Biphenyl-2-Carboxamides, Processes For Their Preparation, Their Use As Medicaments, And Pharmaceutical Preparations Comprising Them SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2009-07-30 US disclosed
US-7514582-B2 2′-substituted 1,1′-biphenyl-2-carboxamides, processes for their preparation, their use as medicaments, and pharmaceutical preparations comprising them SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2009-04-07 US disclosed
US-20040102513-A1 2'-Substituted 1,1'-biphenyl-2-carboxamides, processes for their preparation, their use as medicaments, and pharmaceutical preparations comprising them AVENTIS PHARMA DEUTSCHLAND GMBH 2004-05-27 US disclosed
US-6686395-B2 THERAPY OF A CARDIAC ARRYTHMIA WHICH CAN BE ELIMINATED BY ACTION POTENTIAL PROLONGATION; POTASSIUM CHANNEL MODULATOR AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-02-03 US disclosed
US-20030171351-A1 2'-substituted 1,1'-biphenyl-2-carboxamides, process for their preparation, their use as medicaments, and pharmaceutical preparations comprising them AVENTIS PHARMA DEUTSCHLAND GMBH 2003-09-11 US disclosed
US-6531495-B1 Potassium channel AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2003-03-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030171351-A1 2'-substituted 1,1'-biphenyl-2-carboxamides, process for their preparation, their use as medicaments, and pharmaceutical preparations comprising them MLLT3, RYR2, KCNH1 KMT2A 1459/4885ALDH1A1 217/4885POLB 3577/4885
US-20090192096-A1 2'-Substituted 1,1'-Biphenyl-2-Carboxamides, Processes For Their Preparation, Their Use As Medicaments, And Pharmaceutical Preparations Comprising Them MLLT3, RYR2, CACNA1E KMT2A 1473/4885ALDH1A1 269/4885POLB 3619/4885
US-20040102513-A1 2'-Substituted 1,1'-biphenyl-2-carboxamides, processes for their preparation, their use as medicaments, and pharmaceutical preparations comprising them MLLT3, RYR2, CACNA1E KMT2A 1498/4885ALDH1A1 213/4885POLB 3613/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.