SCHEMBL4246908

SCHEMBL4246908

O=C(O)NCCC=C(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
HPGD P15428 3/20 0.44
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
AKR1B1 P15121 1/20 0.44
GAA P10253 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
ATM Q13315 1/20 0.42
CYP2C9 P11712 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
CNR1 P21554 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
EPHX2 P34913 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL320807 0.74 HPGD (0.68) ALDH1A1HPGDGAAMEN1KMT2A
SCHEMBL10962854 0.73 VNN1 (0.56) ALDH1A1HPGDCES2CES1AKR1B1
SCHEMBL8667929 0.72 CES1 (0.41) ALDH1A1CES2CES1AKR1B1MEN1
Phenethylcarbamic Acid SCHEMBL249525 0.71 CA12 (0.68) ALDH1A1HPGDHDAC8HDAC6TAAR1
SCHEMBL3718010 0.70 ATM (0.60) ALDH1A1HPGDCES2CES1AKR1B1
SCHEMBL11279082 0.70 HPGD (0.62) ALDH1A1HPGDGAAMEN1KMT2A
Phenethylcarbamic Acid SCHEMBL9718519 0.70 CA12 (0.66) ALDH1A1HPGDHDAC8HDAC6TAAR1
Phenethylcarbamic Acid SCHEMBL28010696 0.70 CA12 (0.66) ALDH1A1HPGDHDAC8HDAC6TAAR1
Phenethylcarbamic Acid SCHEMBL4459966 0.70 CA12 (0.66) ALDH1A1HPGDHDAC8HDAC6TAAR1
SCHEMBL28439388 0.69 AKR1B1 (0.48) CES2CES1AKR1B1GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP disclosed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO disclosed