SCHEMBL4254441

SCHEMBL4254441

O=C(C1CCN(C2CN(C(c3ccccc3)c3ccccc3)C2)CC1)N1CCOCC1.O=C(C1CCNCC1)N1CCOCC1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
CNR1 P21554 4/20 0.49
CNR2 P34972 4/20 0.49
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
HTT P42858 2/20 0.47
KDM4E B2RXH2 2/20 0.44
MAPT P10636 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
PIK3CD O00329 1/20 0.42
PIK3CB P42338 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
LMNA P02545 1/20 0.42
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
ACACB O00763 1/20 0.41
ACACA Q13085 1/20 0.41
OPRD1 P41143 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL494586 0.94 ALDH1A1 (0.59) ALDH1A1CNR1CNR2MEN1KMT2A
SCHEMBL4563297 0.92 ALDH1A1 (0.52) ALDH1A1CNR1CNR2MEN1KMT2A
SCHEMBL493765 0.83 ALDH1A1 (0.63) ALDH1A1CNR1CNR2MEN1KMT2A
SCHEMBL3772656 0.81 ALDH1A1 (0.74) ALDH1A1CNR1CNR2KMT2AHTT
SCHEMBL493687 0.77 L3MBTL1 (0.51) ALDH1A1CNR1CNR2KMT2AKDM4E
SCHEMBL6948721 0.76 L3MBTL3 (0.53) ALDH1A1MEN1KMT2AKDM4E
SCHEMBL493492 0.75 TDP1 (0.52) ALDH1A1CNR1CNR2MEN1KMT2A
SCHEMBL693969 0.74 KMT2A (0.66) MEN1KMT2ACYP2C9CYP2C19OPRD1
SCHEMBL493454 0.74 CHRNB2 (0.62) ALDH1A1MEN1KMT2AHTTPIK3CD
Hydrochloric Acid SCHEMBL2591580 0.72 CHRNB2 (0.60) ALDH1A1MEN1KMT2AHTTPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024354-A1 1- [ (4- [BENZOYL (METHYL) AMINO]-3- (PHENYL) BUTYL]AZETIDINE DERIVATIVES FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS 1 Albireo AB (SE) 2009-02-18 EP disclosed
WO-2007136324-A1 1- [ (4- [BENZOYL (METHYL) AMINO] -3- (PHENYL) BUTYL] AZETIDINE DERIVATIVES FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS 1 ALBIREO AB (SE) 2007-11-29 WO disclosed