SCHEMBL4255218

SCHEMBL4255218

CC(C)N1CCN(c2ccc(N)cc2)C(=O)C1.CC(C)N1CCN(c2ccc([N+](=O)[O-])cc2)C(=O)C1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
MAPT P10636 4/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
SIRT6 Q8N6T7 2/20 0.40
ESR1 P03372 2/20 0.39
CYP19A1 P11511 2/20 0.39
ESR2 Q92731 2/20 0.39
KDM4E B2RXH2 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CTSG P08311 1/20 0.38
CMA1 P23946 1/20 0.38
ESRRG P62508 1/20 0.38
KCNJ1 P48048 1/20 0.38
KCNH2 Q12809 1/20 0.38
POLB P06746 1/20 0.38
ADRB1 P08588 1/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4079481 0.95 SIRT6 (0.44) ALDH1A1MAPTMEN1KMT2ASIRT6
SCHEMBL3973870 0.88 HRH3 (0.41) ALDH1A1MAPTMEN1KMT2AESR2
SCHEMBL4256391 0.80 ALDH1A1 (0.47) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL3971995 0.80 ALDH1A1 (0.52) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL854112 0.76 SIRT6 (0.59) ALDH1A1MAPTMEN1KMT2ASIRT6
SCHEMBL23176630 0.76 LMNA (0.44) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL17108484 0.76 MAPT (0.49) ALDH1A1MAPTKDM4ETDP1POLB
SCHEMBL13256438 0.74 NPC1 (0.50) MAPTMEN1KMT2AKDM4ETDP1
SCHEMBL7832831 0.74 SIRT6 (0.38) ALDH1A1MAPTMEN1KMT2ASIRT6
SCHEMBL374834 0.73 SIRT6 (0.68) ALDH1A1MAPTMEN1KMT2ASIRT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907385-A4 COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2009-05-06 EP disclosed
EP-1907385-A2 COMPOUNDS SmithKline Beecham Corporation (US) 2008-04-09 EP disclosed
WO-2007018941-A2 PYRIMIDYL-THIOPHENE DERIVATIVES SMITHKLINE BEECHAM CORPORATION (US) 2007-02-15 WO disclosed