SCHEMBL4258159

SCHEMBL4258159

CC1=C(C(=O)OCc2ccccc2)C(c2ccc3ccccc3c2)c2c(C)n[nH]c2N1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1C Q14123 3/20 0.57
CACNA1B Q00975 1/20 0.54
POLB P06746 1/20 0.47
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
MEN1 O00255 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
MAPT P10636 1/20 0.46
TSHR P16473 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
BRD4 O60885 1/20 0.46
BRD2 P25440 1/20 0.46
BRD3 Q15059 1/20 0.46
BRDT Q58F21 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3004824 0.87 PDE1C (0.69) PDE1CCACNA1BPOLBCYP3A4CYP2C9
SCHEMBL3241017 0.83 PDE1C (0.59) PDE1CCACNA1BPOLBCYP3A4CYP2C9
SCHEMBL2999858 0.75 KDM4E (0.65) CACNA1BPOLBCYP3A4CYP2C9CYP2C19
SCHEMBL10830286 0.74 PDE1C (0.70) PDE1CCACNA1BKDM4EALDH1A1TSHR
SCHEMBL3248414 0.72 MAPT (0.57) CYP3A4CYP2C9CYP2C19KDM4EALDH1A1
SCHEMBL11824598 0.71 ADORA3 (0.73) PDE1CPOLBCYP3A4CYP2C9CYP2C19
SCHEMBL13088047 0.71 PDE1C (0.61) PDE1CCACNA1BKDM4EALDH1A1GAA
SCHEMBL3010323 0.71 MAPT (0.43) PDE1CCACNA1BMAPTBRD4BRD2
SCHEMBL3247037 0.70 ALDH1A1 (0.71) PDE1CPOLBALDH1A1GAAMAPT
SCHEMBL3059809 0.70 GAA (0.73) PDE1CCACNA1BKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009006580-A1 OPTIONALLY CONDENSED DIHYDROPYRIDINE, DIHYDROPYRIMIDINE AND DIHYDROPYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2009-01-08 WO disclosed