SCHEMBL4262821

SCHEMBL4262821

O=P(O)(O)C(Cn1cnc2ncncc21)P(=O)(O)O

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FDPS P14324 8/20 0.62
GGPS1 O95749 3/20 0.54
HDAC6 Q9UBN7 3/20 0.51
HDAC1 Q13547 2/20 0.51
LTA4H P09960 1/20 0.39
HPRT1 P00492 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3976006 0.77 FDPS (1.00) FDPSGGPS1HDAC6HDAC1LTA4H
SCHEMBL13044929 0.76 HDAC6 (0.47) FDPSHDAC6HDAC1LTA4H
SCHEMBL3977299 0.72 FDPS (0.63) FDPSGGPS1HDAC6HDAC1CYP3A4
SCHEMBL30013008 0.72 HDAC6 (0.47) FDPSHDAC6HDAC1LTA4HCYP3A4
SCHEMBL338773 0.72 HDAC6 (0.52) FDPSHDAC6HDAC1LTA4H
SCHEMBL48336 0.71 ADORA2A (0.47) FDPSHDAC6HDAC1LTA4H
SCHEMBL20385726 0.70 FDPS (1.00) FDPSGGPS1HDAC6HDAC1CYP3A4
SCHEMBL3671304 0.68 LTA4H (0.50) HDAC6HDAC1LTA4H
SCHEMBL11066170 0.68 ADORA2A (0.50) HDAC6HDAC1LTA4H
SCHEMBL12472644 0.68 HDAC6 (1.00) HDAC6HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009056952-A1 GEMINAL BISPHOSPHONATES, THEIR PREPARATION AND THEIR USE IN THE FIELD OF ONCOLOGY TETRAPHARM S.R.L. (IT) 2009-05-07 WO claimed
WO-2009056952-A1 GEMINAL BISPHOSPHONATES, THEIR PREPARATION AND THEIR USE IN THE FIELD OF ONCOLOGY TETRAPHARM S.R.L. (IT) 2009-05-07 WO disclosed