SCHEMBL4266773

SCHEMBL4266773

CCOC(=O)c1cccc(N2CC3CNCCN3C2=O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.49
ATM Q13315 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
LMNA P02545 2/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX15 P16050 1/20 0.41
PRKCA P17252 1/20 0.41
GSK3B P49841 1/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
F10 P00742 2/20 0.39
F2 P00734 1/20 0.39
HPN P05981 1/20 0.39
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39
PRSS3 P35030 1/20 0.39
HGFAC Q04756 1/20 0.39
ST14 Q9Y5Y6 1/20 0.39
KHK P50053 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3593426 0.99 ALOX5 (0.48) ALOX5ATMSMN1; SMN2LMNAALDH1A1
SCHEMBL4264273 0.87 ALDH1A1 (0.44) SMN1; SMN2LMNAALDH1A1
SCHEMBL30557800 0.87 ALDH1A1 (0.44) SMN1; SMN2LMNAALDH1A1
Hydrochloric Acid SCHEMBL3607612 0.86 ALDH1A1 (0.43) SMN1; SMN2LMNAALDH1A1
Hydrochloric Acid SCHEMBL3603512 0.84 ALOX5 (0.43) ALOX5LMNAALDH1A1HTR2AHTR2C
SCHEMBL17062844 0.84 ALDH1A1 (0.49) SMN1; SMN2ALDH1A1HTR2CF10F2
SCHEMBL3601344 0.82 HTR2A (0.49) ALOX5HTR2AHTR2CHTR2BF10
Hydrochloric Acid SCHEMBL3602862 0.81 HTR2A (0.48) ALOX5HTR2AHTR2CHTR2BF10
SCHEMBL3597573 0.80 ADRB1 (0.48) ALOX5HTR2AHTR2CHTR2BKHK
Hydrochloric Acid SCHEMBL3603535 0.79 ADRB1 (0.47) ALOX5HTR2AHTR2CHTR2BKHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2039695-A1 BICYCLIC HETEROCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-03-25 EP disclosed