SCHEMBL4264273

SCHEMBL4264273

CCOC(=O)c1ccc(N2CC3CNCCN3C2=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
HTT P42858 5/20 0.44
HPGD P15428 3/20 0.44
NPSR1 Q6W5P4 2/20 0.44
HSP90AA1 P07900 1/20 0.44
CACNA1B Q00975 1/20 0.44
APBA1 Q02410 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 2/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
ALOX12 P18054 1/20 0.41
RECQL P46063 1/20 0.41
KMT2A Q03164 1/20 0.41
IDO1 P14902 1/20 0.41
TSHR P16473 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30557800 1.00 ALDH1A1 (0.44) ALDH1A1HTTHPGDNPSR1HSP90AA1
Hydrochloric Acid SCHEMBL3607612 0.99 ALDH1A1 (0.43) ALDH1A1HTTHPGDNPSR1HSP90AA1
SCHEMBL4266773 0.87 ALOX5 (0.49) ALDH1A1LMNASMN1; SMN2
Hydrochloric Acid SCHEMBL3593426 0.86 ALOX5 (0.48) ALDH1A1LMNASMN1; SMN2
SCHEMBL20941498 0.83 L3MBTL1 (0.42) ALDH1A1MEN1KMT2A
SCHEMBL21863867 0.83 MMP2 (0.44) ALDH1A1HPGDHSD17B10MAPTMEN1
Hydrochloric Acid SCHEMBL22390475 0.82 ALDH1A1 (0.41) ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL22390476 0.82 ALDH1A1 (0.41) ALDH1A1MEN1KMT2A
SCHEMBL17062498 0.82 ALDH1A1 (0.44) ALDH1A1HSD17B10KDM4EUSP2TSHR
SCHEMBL21413824 0.82 ALDH1A1 (0.44) ALDH1A1HSD17B10KDM4EUSP2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2039695-A1 BICYCLIC HETEROCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-03-25 EP disclosed