SCHEMBL4273945

SCHEMBL4273945

O=C(O)/C=C/C1=C(Cc2ccccc2)c2ccccc2CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MITF O75030 1/20 0.47
HSP90AA1 P07900 1/20 0.47
RAB9A P51151 1/20 0.47
ALOX5 P09917 1/20 0.38
LMNA P02545 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
NOTUM Q6P988 1/20 0.38
HDAC3 O15379 1/20 0.38
TNKS O95271 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HCAR2 Q8TDS4 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4270374 1.00 MITF (0.47) MITFHSP90AA1RAB9AALOX5LMNA
Pyrrolidine SCHEMBL4264339 0.92 MITF (0.41) MITFHSP90AA1RAB9AALOX5LMNA
SCHEMBL4274751 0.84 MEN1 (0.45) RAB9ALMNAALDH1A1KDM4EHPGD
SCHEMBL4273001 0.84 CYP1A2 (0.37) MITFHSP90AA1RAB9ALMNAALDH1A1
SCHEMBL4271075 0.84 LMNA (0.42) MITFHSP90AA1RAB9ALMNAALDH1A1
SCHEMBL4264444 0.81 ALDH1A1 (0.44) LMNAALDH1A1KDM4EHPGDMAPK1
SCHEMBL4264446 0.81 ALDH1A1 (0.44) LMNAALDH1A1KDM4EHPGDMAPK1
SCHEMBL4266209 0.79 EGFR (0.55) LMNAHPGDHDAC3HDAC4HDAC1
SCHEMBL4551139 0.77 ESR1 (0.50) MITFHSP90AA1RAB9ALMNAALDH1A1
SCHEMBL4264174 0.77 ESR1 (0.50) MITFHSP90AA1RAB9ALMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110002-A1 NOVEL EFFLUX PUMP INHIBITORS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-09-11 WO disclosed