SCHEMBL4278599

SCHEMBL4278599

Cc1ccc(COc2c(I)cc(C(=O)O)cc2I)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.50
THRB P10828 1/20 0.50
RXRA P19793 3/20 0.48
RXRB P28702 3/20 0.48
MAOB P27338 2/20 0.48
PARP10 Q53GL7 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
TPMT P51580 1/20 0.46
NR1H4 Q96RI1 2/20 0.46
KDM5A P29375 1/20 0.46
KDM2B Q8NHM5 1/20 0.46
KDM4C Q9H3R0 1/20 0.46
KDM5B Q9UGL1 1/20 0.46
RXRG P48443 1/20 0.46
XDH P47989 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
NPC1 O15118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4265171 0.88 RXRA (0.62) RXRARXRBMEN1KMT2ATPMT
SCHEMBL4269670 0.86 MEN1 (0.63) THRATHRBRXRARXRBMEN1
SCHEMBL6731785 0.85 NR4A2 (0.59) RXRARXRBMAOBMEN1KMT2A
SCHEMBL6720945 0.85 NR4A2 (0.59) RXRARXRBMAOBPARP10MEN1
SCHEMBL4274343 0.85 RXRA (0.59) RXRARXRBMAOBMEN1KMT2A
SCHEMBL5014148 0.84 RXRA (0.62) RXRARXRBMEN1KMT2ATPMT
SCHEMBL4275299 0.84 MAOB (0.53) THRATHRBMAOBMEN1KMT2A
SCHEMBL29319558 0.81 RXRA (0.62) RXRARXRBRXRGNPC1POLB
SCHEMBL4265195 0.81 KDM5A (0.49) RXRARXRBMAOBMEN1KMT2A
SCHEMBL6725141 0.81 RXRA (0.55) RXRARXRBMAOBKDM5AKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2066362-A1 RADIOPAQUE AMIDE POLYMERS AND MEDICAL DEVICES FORMED THEREOF Boston Scientific Limited (BB) 2009-06-10 EP claimed
WO-2008033198-A1 RADIOPAQUE AMIDE POLYMERS AND MEDICAL DEVICES FORMED THEREOF BOSTON SCIENTIFIC LIMITED (BB) 2008-03-20 WO claimed
US-20080064848-A1 Radiopaque amide polymers and medical devices formed thereof BOSTON SCIENTIFIC SCIMED, INC. (US) 2008-03-13 US claimed
US-6638977-B1 Biaryl and benzyl ethers and thioethers CORVAS INTERNATIONAL, INC. 2003-10-28 US claimed
WO-2001036351-A2 PLASMINOGEN ACTIVATOR INHIBITOR ANTAGONISTS RELATED APPLICATIONS CORVAS INTERNATIONAL, INC. (US) 2001-05-25 WO claimed
US-8507639-B2 Polyamide block polymers containing iodoarylcarboxyl pendant groups and modified poly(meth)acrylamide; coupling; for tracking movement of a catheter through the body or inflation of balloon at site BOSTON SCIENTIFIC SCIMED, INC. (US) 2013-08-13 US disclosed
US-20080064848-A1 Radiopaque amide polymers and medical devices formed thereof BOSTON SCIENTIFIC SCIMED, INC. (US) 2008-03-13 US disclosed
US-6677473-B1 TREATMENT, PREVENTION OR AMELIORATION OF ONE OR MORE SYMPTOMS OF THROMBOTIC DISORDERS, UNSTABLE ANGINA OR CANCER CORVAS INTERNATIONAL INC 2004-01-13 US disclosed
WO-2001036351-A2 PLASMINOGEN ACTIVATOR INHIBITOR ANTAGONISTS RELATED APPLICATIONS CORVAS INTERNATIONAL, INC. (US) 2001-05-25 WO disclosed