SCHEMBL4279482

SCHEMBL4279482

N=C(NO)c1ccc2c(c1)CCN2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.51
DRD4 P21917 1/20 0.51
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 2/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
CYP2C19 P33261 1/20 0.40
PLAU P00749 1/20 0.39
CRBN Q96SW2 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29673233 0.79 DRD2 (0.55) DRD2DRD4MAPTKDM4EALDH1A1
SCHEMBL773532 0.75 PNMT (0.53) DRD2
SCHEMBL772708 0.75 ASIC3 (0.53) DRD2PLAUF2
SCHEMBL29530477 0.74 KDM4E (0.81) DRD2DRD4MAPTKDM4EALDH1A1
SCHEMBL2638095 0.74 KDM4E (0.81) DRD2DRD4MAPTKDM4EALDH1A1
SCHEMBL2610325 0.72 MAPT (0.58) DRD2DRD4MAPTKDM4EALDH1A1
Hydrochloric Acid SCHEMBL698487 0.72 KDM4E (0.78) DRD2DRD4MAPTKDM4EALDH1A1
SCHEMBL29779540 0.72 KDM4E (0.58) DRD2DRD4MAPTKDM4EALDH1A1
SCHEMBL4051485 0.72 KDM4E (0.58) DRD2DRD4MAPTKDM4EALDH1A1
SCHEMBL18175179 0.72 DRD2 (0.55) DRD2DRD4MAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009151621-A1 SUBSTITUTED (1, 2, 4-0XADIAZ0L-3-YL) INDOLIN-1-YL CARBOXYLIC ACID DERIVATIVES USEFUL AS S1P1 AGONISTS ARENA PHARMACEUTICALS, INC. (US) 2009-12-17 WO disclosed