Alendronic Acid

Alendronic Acid

SCHEMBL4279504

NCCCC(O)(P(=O)(O)O)P(=O)(O)O.[CaH2].[NaH]

nearest known ligand 0.91

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

FDPS

The experimentally established mechanism targets of Alendronic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FDPS known ✓ P14324 17/20 0.91
PDE3A Q14432 3/20 0.91
LMNA P02545 2/20 0.67
ADRB3 P13945 1/20 0.67
PDE4D Q08499 1/20 0.67
GGPS1 O95749 7/20 0.54
CYP3A4 P08684 1/20 0.41
NFKB1 P19838 1/20 0.41
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
AGTR1 P30556 1/20 0.39
OPRM1 P35372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alendronic Acid SCHEMBL6756474 0.98 FDPS (0.87) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL8734225 0.98 FDPS (0.95) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL6856868 0.98 FDPS (0.95) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL1115700 0.98 FDPS (0.95) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL140618 0.98 FDPS (0.95) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL4279497 0.98 FDPS (0.95) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL5974139 0.98 FDPS (0.95) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL140619 0.98 FDPS (0.95) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL192828 0.95 FDPS (0.91) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL579003 0.95 FDPS (0.91) FDPSPDE3ALMNAADRB3PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112316153-B Antitumor pharmaceutical composition and application thereof 中山大学附属第七医院(深圳) 2023-08-25 CN claimed
CN-114349786-B Alam calcium phosphonate super-long nanowire and preparation method and application thereof 中国科学院上海硅酸盐研究所 2023-07-11 CN claimed
CN-114349786-A Alendronate calcium ultralong nanowire and preparation method and application thereof 中国科学院上海硅酸盐研究所 2022-04-15 CN claimed
CN-112707934-A Alendronate calcium complex and preparation method thereof 华南理工大学 2021-04-27 CN claimed
CN-112316153-A Anti-tumor pharmaceutical composition and application thereof 中山大学附属第七医院(深圳) 2021-02-05 CN claimed
US-8974801-B2 Long term sustained release pharmaceutical composition containing aqueous suspension of bisphosphonate AMPHASTAR PHARMACEUTICALS INC. (US) 2015-03-10 US claimed
US-20080011613-A1 Method of electrolytically depositing a pharmaceutical coating onto a conductive osteal implant UNIVERSITY OF BRITISH COLUMBIA, THE (CA) 2008-01-17 US claimed
WO-2006007730-A1 METHOD OF ELECTROLYTICALLY DEPOSITING A PHARMACEUTICAL COATING ONTO A CONDUCTIVE OSTEAL IMPLANT THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2006-01-26 WO claimed
EP-0831756-A1 BISPHOSPHONATE CEMENT COMPOSITION TO PREVENT ASEPTIC LOOSENING OF ORTHOPEDIC IMPLANT DEVICES Merck & Co., Inc. (US) 1998-04-01 EP claimed
WO-1996039107-A1 BISPHOSPHONATE CEMENT COMPOSITION TO PREVENT ASEPTIC LOOSENING OF ORTHOPEDIC IMPLANT DEVICES MERCK & CO., INC. (US) 1996-12-12 WO claimed
CN-112316153-B Antitumor pharmaceutical composition and application thereof 中山大学附属第七医院(深圳) 2023-08-25 CN disclosed
CN-114349786-B Alam calcium phosphonate super-long nanowire and preparation method and application thereof 中国科学院上海硅酸盐研究所 2023-07-11 CN disclosed
CN-114349786-B Alam calcium phosphonate super-long nanowire and preparation method and application thereof 中国科学院上海硅酸盐研究所 2023-07-11 CN disclosed
CN-111544655-B Bisphosphonate type self-coagulation composite bone graft and preparation method thereof 中鼎凯瑞科技成都有限公司 2022-06-24 CN disclosed
CN-114349786-A Alendronate calcium ultralong nanowire and preparation method and application thereof 中国科学院上海硅酸盐研究所 2022-04-15 CN disclosed
US-5589691-A Process for recovery and recycle of methanesulfonic acid and phosphorous acid MERCK & CO., INC. (US) 1996-12-31 US disclosed
WO-1996039107-A1 BISPHOSPHONATE CEMENT COMPOSITION TO PREVENT ASEPTIC LOOSENING OF ORTHOPEDIC IMPLANT DEVICES MERCK & CO., INC. (US) 1996-12-12 WO disclosed
WO-1995033755-A1 PROCESS FOR REMOVING WASTE POx, ALENDRONATE AND ITS BY-PRODUCTS MERCK & CO., INC. (US) 1995-12-14 WO disclosed
WO-1995033756-A1 PROCESS FOR RECOVERY AND RECYCLE OF METHANESULFONIC ACID AND PHOSPHOROUS ACID MERCK & CO., INC. (US) 1995-12-14 WO disclosed
US-5449819-A Process for removing waste pox, alendronate and its by products MERCK & CO., INC. (US) 1995-09-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080011613-A1 Method of electrolytically depositing a pharmaceutical coating onto a conductive osteal implant SOST, CACNA2D1, CACNA2D3 FDPS 2307/4885PDE3A 789/4885LMNA 2694/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.