Alendronic Acid

Alendronic Acid

SCHEMBL192828

NCCCC(O)(P(=O)(O)O)P(=O)(O)O.O.O.O.[NaH]

nearest known ligand 0.91

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

FDPS

The experimentally established mechanism targets of Alendronic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FDPS known ✓ P14324 17/20 0.91
PDE3A Q14432 3/20 0.91
LMNA P02545 2/20 0.67
ADRB3 P13945 1/20 0.67
PDE4D Q08499 1/20 0.67
GGPS1 O95749 7/20 0.54
CYP3A4 P08684 1/20 0.41
NFKB1 P19838 1/20 0.41
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
AGTR1 P30556 1/20 0.39
OPRM1 P35372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alendronic Acid SCHEMBL5973522 1.00 FDPS (0.91) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL7831398 1.00 FDPS (0.91) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL6743637 1.00 FDPS (0.91) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL5974480 1.00 FDPS (0.91) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL1268401 1.00 FDPS (0.91) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL1130855 1.00 FDPS (0.91) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL5973509 1.00 FDPS (0.91) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL1268399 1.00 FDPS (0.91) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL6756474 0.98 FDPS (0.87) FDPSPDE3ALMNAADRB3PDE4D
Alendronic Acid SCHEMBL7751950 0.98 FDPS (0.87) FDPSPDE3ALMNAADRB3PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1188 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116139333-B Carbon fiber reinforced polyether-ether-ketone composite material and preparation method and application thereof 吉林大学 2024-04-12 CN claimed
CN-116139333-A Carbon fiber reinforced polyether-ether-ketone composite material and preparation method and application thereof 吉林大学 2023-05-23 CN claimed
US-20220242893-A1 AMIDE-LINKED CONJUGATE COMPOUNDS AND USES THEREOF UNIV FRASER SIMON (CA) 2022-08-04 US claimed
US-11312737-B2 Amide-linked EP4 agonist-bisphosphonate compounds and uses thereof SIMON FRASER UNIVERSITY (CA) 2022-04-26 US claimed
CN-114306626-A Allan phosphonic acid modified astragaloside IV PEG-PLGA nano micelle and research on anti-osteoporosis effect thereof 席焱海 2022-04-12 CN claimed
US-9592195-B2 Stable effervescent bisphosphonate formulations with rapid solubilization characteristics EFFRX PHARMACEUTICALS SA (CH) 2017-03-14 US claimed
US-9593114-B2 Fluorinated 3-(2-oxo-3-(3-arylpropyl)imidazolidin-1-yl)-3-arylpropanoic acid derivatives SCIFLUOR LIFE SCIENCES, INC. (US) 2017-03-14 US claimed
US-20160130270-A1 FLUORINATED 3-(2-OXO-3-(3-ARYLPROPYL)IMIDAZOLIDIN-1-YL)-3-ARYLPROPANOIC ACID DERIVATIVES FELIQS CORPORATION (JP) 2016-05-12 US claimed
EP-2561877-A1 A Composition containing a Bisphosphonic Acid in combination with Vitamin D Mylan Pharmaceuticals ULC (CA) 2013-02-27 EP claimed
EP-1252162-B1 ALPHA V INTEGRIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2012-07-25 EP claimed
WO-1999030713-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO claimed
WO-1999030709-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO claimed
WO-1999031061-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO claimed
US-5914099-A Prevention of tooth loss by the administration of alendronate or its salts MERCK & CO., INC. (US) 1999-06-22 US claimed
WO-1999004773-A2 METHOD FOR INHIBITING BONE RESORPTION MERCK & CO., INC. (US) 1999-02-04 WO claimed
WO-1998031359-A1 INTEGRIN ANTAGONISTS MERCK & CO., INC. (US) 1998-07-23 WO claimed
WO-1998014196-A1 LIQUID ALENDRONATE FORMULATIONS MERCK & CO., INC. (US) 1998-04-09 WO claimed
EP-0824341-A1 PREVENTION OF TOOTH LOSS BY THE ADMINISTRATION OF ALENDRONATE OR ITS SALTS Merck & Co., Inc. (US) 1998-02-25 EP claimed
US-5646134-A INHIBITING BONE RESORPTION MERCK & CO., INC. (US) 1997-07-08 US claimed
WO-1996035407-A1 PREVENTION OF TOOTH LOSS BY THE ADMINISTRATION OF ALENDRONATE OR ITS SALTS MERCK & CO., INC. (US) 1996-11-14 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160130270-A1 FLUORINATED 3-(2-OXO-3-(3-ARYLPROPYL)IMIDAZOLIDIN-1-YL)-3-ARYLPROPANOIC ACID DERIVATIVES ITGB3, ITGA2, ITGA1 FDPS 1908/4885PDE3A 2026/4885LMNA 2972/4885
US-11312737-B2 Amide-linked EP4 agonist-bisphosphonate compounds and uses thereof PTGER4, ENPP2, GPR4 FDPS 1484/4885PDE3A 1505/4885LMNA 3845/4885
US-20220242893-A1 AMIDE-LINKED CONJUGATE COMPOUNDS AND USES THEREOF AADAC, DNPEP, NAALAD2 FDPS 769/4885PDE3A 2015/4885LMNA 3003/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.