SCHEMBL4282428

SCHEMBL4282428

N#Cc1ccc(-c2n[nH]cc2-c2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.46
KDM1A O60341 1/20 0.46
MAPK13 O15264 1/20 0.46
RAF1 P04049 1/20 0.46
MAPK12 P53778 1/20 0.46
MAPK11 Q15759 1/20 0.46
MAPK14 Q16539 1/20 0.46
ERBB2 P04626 2/20 0.45
GRM5 P41594 2/20 0.43
TSHR P16473 1/20 0.42
GABRA1 P14867 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42
MAOA P21397 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.41
CYP11B2 P19099 1/20 0.41
TDO2 P48775 1/20 0.40
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30239600 0.86 MAPK14 (0.49) KDM1AMAPK13RAF1MAPK12MAPK11
SCHEMBL218119 0.84 ALOX15 (0.52) ERBB2GRM5IDO1NPC1RAB9A
SCHEMBL24963519 0.79 AURKA (0.45) MAOBMAPK13RAF1MAPK12MAPK11
SCHEMBL28329372 0.77 ADORA1 (0.49) MAPK13MAPK12MAPK11MAPK14ADORA1
SCHEMBL1128951 0.77 ALDH1A1 (0.50) MAPK13MAPK12MAPK11MAPK14ERBB2
SCHEMBL1129154 0.77 ALDH1A1 (0.50) MAPK13MAPK12MAPK11MAPK14ERBB2
SCHEMBL3108967 0.77 TDP1 (0.52) NPC1RAB9AADORA1
SCHEMBL28197453 0.76 ALOX15 (0.43) GRM5IDO1RAB9AADORA1
SCHEMBL1847072 0.76 CLK4 (0.45) MAOBMAPK14GRM5CYP11B2TDO2
SCHEMBL27844934 0.76 ERBB2 (0.41) MAOBKDM1AMAPK13RAF1MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009151991-A1 PYRAZOLE DERIVATIVES USEFUL AS INHIBITORS OF FAAH MERCK & CO., INC. (US) 2009-12-17 WO disclosed