SCHEMBL4282666

SCHEMBL4282666

COc1ccccc1CC(Br)C(C)=O

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.50
MTNR1B P49286 1/20 0.50
ALDH1A1 P00352 4/20 0.47
HPGD P15428 3/20 0.47
HTT P42858 1/20 0.47
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
TSHR P16473 1/20 0.43
IDO1 P14902 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
GAA P10253 1/20 0.43
POLB P06746 1/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6695813 0.83 MTNR1A (0.53) MTNR1AMTNR1BALDH1A1HPGDHTT
SCHEMBL14250613 0.81 MTNR1A (0.51) MTNR1AMTNR1BALDH1A1HPGDHTT
SCHEMBL17478028 0.80 MTNR1A (0.50) MTNR1AMTNR1BALDH1A1HPGDHTT
SCHEMBL17670826 0.79 ALDH1A1 (0.49) MTNR1AMTNR1BALDH1A1HPGDHTT
SCHEMBL9480529 0.78 IDO1 (0.52) MTNR1AMTNR1BALDH1A1HPGDHTT
SCHEMBL28805376 0.78 IDO1 (0.52) ALDH1A1MEN1KMT2AIDO1TAAR1
SCHEMBL27942554 0.78 MTNR1A (0.51) MTNR1AMTNR1BALDH1A1HPGDHTT
SCHEMBL7385695 0.76 CYP1A2 (0.59) MTNR1AMTNR1BALDH1A1HPGDHTT
SCHEMBL6206375 0.75 IDO1 (0.48) MTNR1AMTNR1BALDH1A1HPGDHTT
SCHEMBL2426744 0.75 ALDH1A1 (0.46) MTNR1AMTNR1BALDH1A1HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed