SCHEMBL4285447

SCHEMBL4285447

CCc1c(C(N)=O)cccc1-c1cc(OC)cc(OC)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.44
TP53 P04637 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
KDM4E B2RXH2 1/20 0.44
RECQL P46063 1/20 0.44
MAPK10 P53779 1/20 0.44
ABL1 P00519 2/20 0.43
ABCB1 P08183 2/20 0.43
BCR P11274 2/20 0.43
AURKA O14965 1/20 0.43
RPS6KB1 P23443 1/20 0.43
AURKB Q96GD4 1/20 0.43
PARP1 P09874 7/20 0.43
PDK2 Q15119 1/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2E1 P05181 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C8 P10632 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28187515 0.82 BCAT2 (0.58) NPC1TP53RAB9ASMN1; SMN2KDM4E
SCHEMBL4439618 0.79 BCAT2 (0.62) NPC1RAB9ASMN1; SMN2PARP1IKBKB
SCHEMBL4285442 0.79 NPC1 (0.45) NPC1TP53RAB9ASMN1; SMN2KDM4E
SCHEMBL5517154 0.77 PARP1 (0.51) NPC1TP53RAB9ASMN1; SMN2PARP1
SCHEMBL45719 0.75 PARP1 (0.51) KDM4EPARP1CYP3A4MAPT
SCHEMBL23647145 0.74 PKN1 (0.46) ABL1PARP1PDK2CDC7IKBKB
SCHEMBL2998004 0.74 SMN1; SMN2 (0.55) TP53SMN1; SMN2KDM4ECYP1A2CYP2D6
SCHEMBL1135994 0.74 CTSD (0.49) NPC1TP53RAB9ASMN1; SMN2PARP1
SCHEMBL4709256 0.74 BCAT2 (0.59) NPC1TP53RAB9ASMN1; SMN2KDM4E
SCHEMBL16463069 0.73 PARP1 (0.44) KDM4EPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1675552-A4 PREPERATION OF 1,6-DISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LTD (GB) 2009-06-03 EP disclosed
EP-1675552-A2 PREPERATION OF 1,6-DISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-07-05 EP disclosed
WO-2005037197-A2 PREPERATION OF 1,6-DISUBSTITUTED AZABENZIMIDAZOLES AS KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2005-04-28 WO disclosed