SCHEMBL4285491

SCHEMBL4285491

CC1C(c2ccc(F)cc2)CCCN1C(=O)ON

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
HRH3 Q9Y5N1 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
HCRTR2 O43614 1/20 0.39
SLC9A1 P19634 1/20 0.38
THRB P10828 1/20 0.38
ALOX12 P18054 1/20 0.38
MEN1 O00255 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
ALDH1A1 P00352 1/20 0.37
SLC6A3 Q01959 3/20 0.37
SLC6A2 P23975 2/20 0.37
NR3C2 P08235 1/20 0.37
SLC6A4 P31645 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4291623 0.86 HCRTR2 (0.41) HCRTR2
SCHEMBL4282511 0.86 HSD17B10 (0.46) KMT2ASMN1; SMN2HCRTR2MEN1MAPK1
SCHEMBL4291881 0.84 SLC6A3 (0.40) HCRTR2ALDH1A1SLC6A3SLC6A2SLC6A4
SCHEMBL4280118 0.84 HTR2A (0.40) HRH3HCRTR2SLC9A1
SCHEMBL4282253 0.82 TACR1 (0.41) HCRTR2
SCHEMBL4292808 0.81 SLC6A3 (0.45) HTTSLC6A3SLC6A2SLC6A4
SCHEMBL4288935 0.80 TSHR (0.39) SMN1; SMN2HTTSLC6A3SLC6A2SLC6A4
SCHEMBL4285848 0.79 SLC6A2 (0.42) HRH3SMN1; SMN2HCRTR2HTTALDH1A1
SCHEMBL4294068 0.79 POLB (0.36) SMN1; SMN2SIGMAR1ALDH1A1
SCHEMBL4285494 0.77 SLC6A3 (0.43) KMT2ATHRBALOX12SLC6A3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009072643-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-11 WO disclosed