SCHEMBL4280118

SCHEMBL4280118

Cc1cc(C2CCCN(C(=O)ON)C2C)ccc1F

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
SLC9A1 P19634 2/20 0.35
HCRTR1 O43613 2/20 0.34
HCRTR2 O43614 2/20 0.34
HSD11B1 P28845 2/20 0.34
BTK Q06187 1/20 0.34
CNR2 P34972 1/20 0.34
GRIN2B Q13224 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
PDE2A O00408 1/20 0.33
HTR7 P34969 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4291881 0.91 SLC6A3 (0.40) HCRTR1HCRTR2HSD11B1
SCHEMBL4291623 0.91 HCRTR2 (0.41) HTR2AHTR2CHTR2BHCRTR2HSD11B1
SCHEMBL4285848 0.86 SLC6A2 (0.42) HCRTR1HCRTR2HSD11B1BTKHRH3
SCHEMBL4288935 0.85 TSHR (0.39) HSD11B1
SCHEMBL4285491 0.84 KMT2A (0.41) SLC9A1HCRTR2HRH3
SCHEMBL4292808 0.81 SLC6A3 (0.45)
SCHEMBL4280120 0.80 LMNA (0.40) HTR2AHTR2CHTR2BSLC9A1HCRTR1
SCHEMBL4294068 0.79 POLB (0.36) HSD11B1BTK
SCHEMBL4282253 0.79 TACR1 (0.41) HCRTR1HCRTR2
SCHEMBL4282511 0.78 HSD17B10 (0.46) HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009072643-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-11 WO disclosed