SCHEMBL4282253

SCHEMBL4282253

Cc1cc(F)ccc1C1CCCN(C(=O)ON)C1C

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.41
OPRL1 P41146 2/20 0.38
HCRTR2 O43614 5/20 0.38
RIPK1 Q13546 1/20 0.37
GRM5 P41594 2/20 0.36
HCRTR1 O43613 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4285491 0.82 KMT2A (0.41) HCRTR2
SCHEMBL4291881 0.79 SLC6A3 (0.40) HCRTR2RIPK1HCRTR1
SCHEMBL4282256 0.79 HCRTR2 (0.43) TACR1OPRL1HCRTR2RIPK1GRM5
SCHEMBL4280118 0.79 HTR2A (0.40) HCRTR2HCRTR1
SCHEMBL4291623 0.76 HCRTR2 (0.41) HCRTR2
SCHEMBL4288935 0.75 TSHR (0.39) NPSR1
SCHEMBL4285848 0.74 SLC6A2 (0.42) HCRTR2HCRTR1
SCHEMBL4281406 0.74 KDM4E (0.36) NPSR1
SCHEMBL4294068 0.72 POLB (0.36)
SCHEMBL4292808 0.71 SLC6A3 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009072643-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-11 WO disclosed