SCHEMBL4285849

SCHEMBL4285849

COC(=O)N1CCCC(c2ccc(Cl)c(C)c2)C1N

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 9/20 0.47
SLC6A3 Q01959 9/20 0.47
SLC6A2 P23975 6/20 0.47
CHRNB4 P30926 4/20 0.47
CHRNA3 P32297 4/20 0.47
CHRNA1 P02708 3/20 0.47
CHRNG P07510 3/20 0.47
ITGA5 P08648 3/20 0.47
CHRNB1 P11230 3/20 0.47
CHRNB2 P17787 3/20 0.47
CHRNA4 P43681 3/20 0.47
CHRND Q07001 3/20 0.47
TSHR P16473 1/20 0.39
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
OPRK1 P41145 2/20 0.38
OPRM1 P35372 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4288939 0.92 TSHR (0.44) SLC6A4SLC6A3SLC6A2CHRNB4CHRNA3
SCHEMBL4292811 0.90 SLC6A4 (0.51) SLC6A4SLC6A3SLC6A2
SCHEMBL4280120 0.86 LMNA (0.40) SLC6A4SLC6A3SLC6A2CHRNB4CHRNA3
SCHEMBL4291883 0.83 SLC6A3 (0.46) SLC6A4SLC6A3SLC6A2CHRNB4CHRNA3
SCHEMBL4294072 0.81 CHRNB4 (0.41) CHRNB4CHRNA3HCRTR1HCRTR2OPRK1
SCHEMBL4291624 0.81 HCRTR2 (0.42) HCRTR2OPRK1
SCHEMBL4285848 0.80 SLC6A2 (0.42) SLC6A4SLC6A3SLC6A2CHRNB4CHRNA3
SCHEMBL4285494 0.79 SLC6A3 (0.43) SLC6A4SLC6A3SLC6A2
SCHEMBL4282512 0.79 HCRTR2 (0.47) SLC6A4SLC6A3SLC6A2TSHRHCRTR2
SCHEMBL4281409 0.77 ALDH1A1 (0.38) ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009072643-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-11 WO disclosed