SCHEMBL4288939

SCHEMBL4288939

COC(=O)N1CCCC(c2ccc(C)c(Cl)c2)C1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.44
MAPT P10636 3/20 0.43
SLC6A2 P23975 5/20 0.42
SLC6A4 P31645 5/20 0.42
SLC6A3 Q01959 5/20 0.42
NPSR1 Q6W5P4 2/20 0.41
LMNA P02545 1/20 0.41
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
CHRNB4 P30926 3/20 0.39
CHRNA3 P32297 3/20 0.39
CHRNA1 P02708 2/20 0.39
CHRNG P07510 2/20 0.39
ITGA5 P08648 2/20 0.39
CHRNB1 P11230 2/20 0.39
CHRNB2 P17787 2/20 0.39
CHRNA4 P43681 2/20 0.39
CHRND Q07001 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4285849 0.92 SLC6A4 (0.47) TSHRSLC6A2SLC6A4SLC6A3CHRNB4
SCHEMBL4292811 0.91 SLC6A4 (0.51) SLC6A2SLC6A4SLC6A3
SCHEMBL4291883 0.87 SLC6A3 (0.46) TSHRMAPTSLC6A2SLC6A4SLC6A3
SCHEMBL4280120 0.84 LMNA (0.40) TSHRMAPTSLC6A2SLC6A4SLC6A3
SCHEMBL4291624 0.84 HCRTR2 (0.42) NPSR1L3MBTL1
SCHEMBL4294072 0.82 CHRNB4 (0.41) CHRNB4CHRNA3SMN1; SMN2ALDH1A1
SCHEMBL4285494 0.80 SLC6A3 (0.43) SLC6A2SLC6A4SLC6A3
SCHEMBL4282512 0.80 HCRTR2 (0.47) TSHRSLC6A2SLC6A4SLC6A3SMN1; SMN2
SCHEMBL4288935 0.80 TSHR (0.39) TSHRMAPTSLC6A2SLC6A4SLC6A3
SCHEMBL4286379 0.78 SLC6A4 (0.47) SLC6A2SLC6A4SLC6A3HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009072643-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-11 WO disclosed