SCHEMBL4289075

SCHEMBL4289075

O=C(O)N1c2ccccc2CC1CO

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.53
DRD4 P21917 1/20 0.53
NOTUM Q6P988 1/20 0.49
NPC1 O15118 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
ACE P12821 3/20 0.45
AKT1 P31749 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30681441 1.00 DRD2 (0.53) DRD2DRD4NOTUMNPC1ALDH1A1
SCHEMBL7554164 1.00 DRD2 (0.53) DRD2DRD4NOTUMNPC1ALDH1A1
SCHEMBL7993369 0.85 DRD2 (0.54) DRD2DRD4NOTUMNPC1ALDH1A1
SCHEMBL3441713 0.84 ACE (0.47) ACE
SCHEMBL30681525 0.81 NOTUM (0.48) NOTUMNPC1ALDH1A1CYP1A2CYP2C19
SCHEMBL4386325 0.81 NOTUM (0.44) NOTUMNPC1ALDH1A1CYP1A2CYP2C19
SCHEMBL30681248 0.80 DRD2 (0.45) DRD2DRD4NOTUMNPC1ALDH1A1
SCHEMBL4436739 0.80 NOTUM (0.43) DRD2DRD4NOTUMACE
SCHEMBL5763420 0.80 NPC1 (0.53) DRD2DRD4NPC1CYP2C19
SCHEMBL24201848 0.79 DRD2 (0.53) DRD2DRD4NOTUMNPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102762567-A Diaza-spiro[5.5]undecanes as orexin receptor antagonists NOVARTIS AG 2012-10-31 CN disclosed
WO-2009151626-A1 SUBSTITUTED (1, 2, 4-0XADIAZ0L-3-YL) INDOLIN-1-YL CARBOXYLIC ACID DERIVATIVES USEFUL AS S1P1 AGONISTS ARENA PHARMACEUTICALS, INC. (US) 2009-12-17 WO disclosed