SCHEMBL4291667

SCHEMBL4291667

CN(C)C(=O)N1CCCC(c2ccc(Cl)c(Cl)c2)C1N

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 5/20 0.45
SLC6A4 P31645 4/20 0.45
SLC6A2 P23975 2/20 0.45
UTS2R Q9UKP6 4/20 0.42
OPRK1 P41145 4/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4292811 0.84 SLC6A4 (0.51) SLC6A3SLC6A4SLC6A2
SCHEMBL4286379 0.83 SLC6A4 (0.47) SLC6A3SLC6A4SLC6A2HTT
SCHEMBL4292808 0.76 SLC6A3 (0.45) SLC6A3SLC6A4SLC6A2UTS2RHTT
SCHEMBL4288939 0.76 TSHR (0.44) SLC6A3SLC6A4SLC6A2HTT
SCHEMBL4285849 0.75 SLC6A4 (0.47) SLC6A3SLC6A4SLC6A2OPRK1
SCHEMBL4288935 0.68 TSHR (0.39) SLC6A3SLC6A4SLC6A2HTT
SCHEMBL4294072 0.67 CHRNB4 (0.41) OPRK1
SCHEMBL4285848 0.67 SLC6A2 (0.42) SLC6A3SLC6A4SLC6A2HTT
SCHEMBL4291624 0.67 HCRTR2 (0.42) OPRK1
SCHEMBL10192778 0.66 SLC6A2 (0.45) SLC6A3SLC6A4SLC6A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009072643-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-11 WO disclosed