SCHEMBL4293828

SCHEMBL4293828

Cn1cc(C(=O)c2cc(Cl)ncn2)c2ccc(C#N)cc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
IMPDH2 P12268 2/20 0.35
NTRK1 P04629 3/20 0.35
HDAC3 O15379 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
KDM1A O60341 1/20 0.35
POLB P06746 1/20 0.35
SCN9A Q15858 2/20 0.35
CACNA1H O95180 1/20 0.35
PGR P06401 1/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CDK1 P06493 1/20 0.34
EDNRA P25101 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3992947 0.86 POLB (0.38) CNR1CNR2NTRK1POLBMEN1
SCHEMBL3992240 0.86 POLB (0.38) CNR1CNR2IMPDH2NTRK1POLB
SCHEMBL3997478 0.84 POLB (0.36) CNR1CNR2POLBMEN1MAPT
SCHEMBL3978572 0.84 PCSK9 (0.40) CNR1CNR2NTRK1POLBMEN1
SCHEMBL3972624 0.82 POLB (0.55) POLBMEN1MAPTKMT2A
SCHEMBL3995936 0.82 ALDH1A1 (0.44) CNR2HDAC3HDAC1HDAC2HDAC8
SCHEMBL3990286 0.81 SCN9A (0.40) CNR1CNR2NTRK1POLBSCN9A
SCHEMBL3996013 0.79 KDR (0.41) CNR1CNR2POLBMEN1MAPT
SCHEMBL3990318 0.78 NR4A2 (0.35) CNR2HDAC3HDAC1HDAC2HDAC8
SCHEMBL3973248 0.77 KDM4E (0.42) CNR1CNR2NTRK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2065382-A1 CGRP antagonists Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2009-06-03 EP disclosed