SCHEMBL4294185

SCHEMBL4294185

CCCCCCCCCCOCC(COCCCCCC)OCCCCCC

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 9/20 0.68
LPAR3 Q9UBY5 9/20 0.68
LPAR2 Q9HBW0 6/20 0.68
DNM1 Q05193 1/20 0.59
USP2 O75604 1/20 0.55
HTT P42858 1/20 0.53
TLR2 O60603 4/20 0.53
PRKD3 O94806 1/20 0.52
PRKCG P05129 1/20 0.52
PRKCB P05771 1/20 0.52
PRKCA P17252 1/20 0.52
PRKCH P24723 1/20 0.52
PRKCI P41743 1/20 0.52
PRKCE Q02156 1/20 0.52
PRKCQ Q04759 1/20 0.52
PRKCZ Q05513 1/20 0.52
PRKCD Q05655 1/20 0.52
PRKD1 Q15139 1/20 0.52
LPAR6 P43657 5/20 0.50
LPAR4 Q99677 5/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7183039 1.00 LPAR1 (0.68) LPAR1LPAR3LPAR2DNM1USP2
SCHEMBL30510651 1.00 LPAR1 (0.68) LPAR1LPAR3LPAR2DNM1USP2
SCHEMBL30910033 1.00 LPAR1 (0.68) LPAR1LPAR3LPAR2DNM1USP2
SCHEMBL30510614 1.00 LPAR1 (0.68) LPAR1LPAR3LPAR2DNM1USP2
SCHEMBL8636551 1.00 LPAR1 (0.68) LPAR1LPAR3LPAR2DNM1USP2
SCHEMBL4204833 1.00 LPAR1 (0.68) LPAR1LPAR3LPAR2DNM1USP2
SCHEMBL303128 1.00 LPAR1 (0.68) LPAR1LPAR3LPAR2DNM1USP2
SCHEMBL7563995 1.00 LPAR1 (0.68) LPAR1LPAR3LPAR2DNM1USP2
SCHEMBL4879843 1.00 LPAR1 (0.68) LPAR1LPAR3LPAR2DNM1USP2
SCHEMBL4204708 1.00 LPAR1 (0.68) LPAR1LPAR3LPAR2DNM1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260071218-A1 Oral Delivery of Antisense Conjugates Targeting PCSK9 CIVI BIOPHARMA INC (US) 2026-03-12 US disclosed
EP-4705454-A2 COMPOUNDS AND METHODS FOR TREATING HUMAN SUBJECTS Stoke Therapeutics, Inc. (US) 2026-03-11 EP disclosed
EP-4705455-A1 COMPOUNDS AND METHODS FOR TREATING HUMAN SUBJECTS Stoke Therapeutics, Inc. (US) 2026-03-11 EP disclosed
US-20260055409-A1 COMPOUNDS AND METHODS FOR TREATING HUMAN SUBJECTS STOKE THERAPEUTICS INC (US) 2026-02-26 US disclosed
US-12421516-B2 Antisense oligomers targeting PCSK9 ROCHE INNOVATION CENTER COPENHAGEN A/S (DK) 2025-09-23 US disclosed
US-12291708-B2 Oral delivery of antisense conjugates targeting PCSK9 CIVI BIOPHARMA, INC. (US) 2025-05-06 US disclosed
WO-2024229421-A1 COMPOUNDS AND METHODS FOR TREATING HUMAN SUBJECTS STOKE THERAPEUTICS, INC. (US) 2024-11-07 WO disclosed
WO-2024227085-A2 COMPOUNDS AND METHODS FOR TREATING HUMAN SUBJECTS STOKE THERAPEUTICS, INC. (US) 2024-10-31 WO disclosed
US-20240084307-A1 ANTISENSE OLIGOMERS TARGETING PCSK9 ROCHE INNOVATION CENTER COPENHAGEN A/S (DK) 2024-03-14 US disclosed
US-20240067965-A1 ORAL DELIVERY OF ANTISENSE CONJUGATES TARGETING PCSK9 CIVI BIOPHARMA INC (US) 2024-02-29 US disclosed
US-7608705-B2 nucleobases are cytosine groups or mimetics; modified with polyethyleneglycol or a tocopheryl group; useful in inhibiting proliferation of pancreatic tumors UNIVERSITATSKLINIKUM SCHLESWIG-HOLSTEIN (DE) 2009-10-27 US disclosed
US-20090203132-A1 PYRROLIDINYL GROUPS FOR ATTACHING CONJUGATES TO OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS, INC. 2009-08-13 US disclosed
US-20080199960-A1 Methods for the Delivery of Oligomeric Compounds K.U. LEUVEN RESEARCH AND DEVELOPMENT (BE) 2008-08-21 US disclosed
WO-2006031461-A2 PYRROLIDINYL GROUPS FOR ATTACHING CONJUGATES TO OLIGOMERIC COMPOUNDS ISIS PHARMACEUTICALS, INC. (US) 2006-03-23 WO disclosed
US-20050119470-A1 Conjugated oligomeric compounds and their use in gene modulation ISIS PHARMACEUTICALS, INC. 2005-06-02 US disclosed
US-20050019761-A1 Oligonucleotides, agents containing these oligonucleotides, and the use thereof UNIVERSITATSKLINIKUM SCHLESWIG-HOLSTEIN (DE) 2005-01-27 US disclosed
WO-2004044141-A2 CONJUGATED OLIGOMERIC COMPOUNDS AND THEIR USE IN GENE MODULATION ISIS PHARMACEUTICALS, INC. (US) 2004-05-27 WO disclosed
EP-1326878-A2 OLIGONUCLEOTIDES, AGENTS CONTAINING THESE OLIGONUCLEOTIDES, AND THE USE THEREOF Bayer, Ernst, Prof. Dr. (DE) 2003-07-16 EP disclosed
WO-2002026754-A9 OLIGONUCLEOTIDES, AGENTS CONTAINING THESE OLIGONUCLEOTIDES, AND THE USE THEREOF BAYER ERNST (DE) 2003-05-15 WO disclosed
WO-2002026754-A2 OLIGONUCLEOTIDES, AGENTS CONTAINING THESE OLIGONUCLEOTIDES, AND THE USE THEREOF BAYER ERNST (DE) 2002-04-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12421516-B2 Antisense oligomers targeting PCSK9 PCSK9, PCSK7, PCSK6 LPAR1 75/4885LPAR3 32/4885LPAR2 106/4885
US-20090203132-A1 PYRROLIDINYL GROUPS FOR ATTACHING CONJUGATES TO OLIGOMERIC COMPOUNDS PHAX, RIOX2, RNMT LPAR1 2494/4885LPAR3 1618/4885LPAR2 1751/4885
US-20260071218-A1 Oral Delivery of Antisense Conjugates Targeting PCSK9 PCSK9, ALPI, SLC10A2 LPAR1 295/4885LPAR3 347/4885LPAR2 236/4885
US-20240067965-A1 ORAL DELIVERY OF ANTISENSE CONJUGATES TARGETING PCSK9 PCSK9, SCD5, PCSK7 LPAR1 540/4885LPAR3 239/4885LPAR2 379/4885
US-20260055409-A1 COMPOUNDS AND METHODS FOR TREATING HUMAN SUBJECTS CYFIP1, SYNGR2, CYFIP2 LPAR1 3026/4885LPAR3 3949/4885LPAR2 3163/4885
US-12291708-B2 Oral delivery of antisense conjugates targeting PCSK9 PCSK9, SCD5, PCSK7 LPAR1 540/4885LPAR3 239/4885LPAR2 379/4885
US-20050119470-A1 Conjugated oligomeric compounds and their use in gene modulation PHAX, SNRPE, RRP1B LPAR1 1902/4885LPAR3 1338/4885LPAR2 1366/4885
US-20240084307-A1 ANTISENSE OLIGOMERS TARGETING PCSK9 PCSK9, PCSK7, PCSK6 LPAR1 75/4885LPAR3 32/4885LPAR2 106/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.