SCHEMBL4296964

SCHEMBL4296964

Nc1ccc(Cl)c(CN2CC(O)C2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.44
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 1/20 0.44
TDP1 Q9NUW8 2/20 0.43
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
BCL2L1 Q07817 1/20 0.43
GBA1 P04062 1/20 0.39
HTT P42858 1/20 0.39
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
P2RX7 Q99572 1/20 0.37
CD274 Q9NZQ7 3/20 0.37
PDCD1LG2 Q9BQ51 2/20 0.37
FAAH O00519 1/20 0.36
CXCR4 P61073 1/20 0.36
PDCD1 Q15116 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4291807 0.81 KMT2A (0.48) ACHEKDM4EALDH1A1LMNAMAPT
SCHEMBL3398877 0.80 VEGFA (0.46) ALDH1A1TDP1MAPTSMN1; SMN2HTT
SCHEMBL13861951 0.78 ACHE (0.65) ACHEKDM4EALDH1A1LMNATDP1
SCHEMBL15065984 0.77 ACHE (0.63) ACHEKDM4EALDH1A1TDP1MAPT
SCHEMBL3110747 0.76 KDM4E (0.63) KDM4EALDH1A1MAPTHTTFAAH
SCHEMBL3396517 0.75 GBA1 (0.61) ALDH1A1LMNAGBA1S1PR1S1PR5
SCHEMBL4297559 0.74 LMNA (0.60) ACHEKDM4EALDH1A1LMNATDP1
SCHEMBL15687883 0.74 ALDH1A1 (0.54) ACHEKDM4EALDH1A1LMNATDP1
SCHEMBL520610 0.74 CYP2A13 (0.61) ACHEKDM4EALDH1A1TDP1MAPT
SCHEMBL4371470 0.73 LTA4H (0.41) ACHEKDM4EALDH1A1LMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8420657-B2 Pyrrolo[2,3-D]pyrimidines and use thereof as tyrosine kinase inhibitors NOVARTIS AG (CH) 2013-04-16 US disclosed
US-20090203688-A1 HETEROCYCLIC COMPOUNDS NOVARTIS AG 2009-08-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090203688-A1 HETEROCYCLIC COMPOUNDS ABL1, JAK2, JAK1 ACHE 4251/4885KDM4E 1741/4885ALDH1A1 1389/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.