SCHEMBL4307202

SCHEMBL4307202

COc1ccc(Cl)cc1NC(=O)N1CCN(CCO)CC1

nearest known ligand 0.77

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.77
RBP4 P02753 6/20 0.70
MAPT P10636 2/20 0.66
LMNA P02545 2/20 0.62
GAA P10253 1/20 0.58
ALDH1A1 P00352 2/20 0.57
KCNT1 Q5JUK3 1/20 0.56
THRB P10828 2/20 0.56
KMT2A Q03164 3/20 0.55
MEN1 O00255 2/20 0.55
POLB P06746 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16690803 0.87 MAPK1 (1.00) MAPK1RBP4MAPTLMNAGAA
SCHEMBL4306582 0.87 MAPT (0.73) MAPK1RBP4MAPTLMNAKCNT1
SCHEMBL4301167 0.82 MAPT (0.67) MAPK1RBP4MAPTLMNAALDH1A1
SCHEMBL16690852 0.82 RBP4 (1.00) MAPK1RBP4MAPTLMNAALDH1A1
Iodide SCHEMBL4152138 0.80 MAPT (0.61) MAPK1RBP4MAPTLMNAGAA
SCHEMBL16690848 0.80 RBP4 (0.83) MAPK1RBP4MAPTLMNAGAA
SCHEMBL27695780 0.79 ROS1 (0.56) MAPK1MAPTALDH1A1POLB
SCHEMBL4451899 0.79 RBP4 (0.67) MAPK1RBP4MAPTLMNAKCNT1
SCHEMBL16690825 0.79 RBP4 (1.00) MAPK1RBP4MAPTLMNAGAA
Iodide SCHEMBL4161671 0.79 MAPT (0.69) MAPK1RBP4MAPTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090118303-A1 SEROTONIN 5-HT3 RECEPTOR AGONIST RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2009-05-07 US disclosed
US-7485646-B2 Serotonin 5-HT3 receptor agonist RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2009-02-03 US disclosed
US-20070265277-A1 Serotonin 5-Ht3 Receptor Agonist RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2007-11-15 US disclosed
EP-1798227-A1 SEROTONIN 5-HT3 RECEPTOR AGONIST Research Foundation Itsuu Laboratory (JP) 2007-06-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090118303-A1 SEROTONIN 5-HT3 RECEPTOR AGONIST HTR3A, HTR7, HTR1A MAPK1 1292/4885RBP4 3590/4885MAPT 4268/4885
US-20070265277-A1 Serotonin 5-Ht3 Receptor Agonist HTR3A, HTR7, HTR1A MAPK1 1292/4885RBP4 3590/4885MAPT 4268/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.