SCHEMBL431501

SCHEMBL431501

Cc1ccc(C(=O)O)c(I)c1[N+](=O)[O-]

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
TDP1 Q9NUW8 3/20 0.46
TSHR P16473 6/20 0.44
CYP3A4 P08684 2/20 0.40
ALOX15 P16050 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PKM P14618 1/20 0.40
POLB P06746 2/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2263102 0.89 TSHR (0.46) ALDH1A1TDP1TSHRCYP3A4ALOX15
SCHEMBL28300921 0.85 TSHR (0.53) ALDH1A1TDP1TSHRCYP3A4ALOX15
SCHEMBL2381586 0.82 TSHR (0.54) ALDH1A1TDP1TSHRCYP3A4ALOX15
SCHEMBL2598195 0.81 TDP1 (0.49) ALDH1A1TDP1TSHRCYP3A4ALOX15
SCHEMBL5314234 0.81 ALDH1A1 (0.47) ALDH1A1TDP1TSHRCYP3A4ALOX15
SCHEMBL1355836 0.80 TSHR (0.51) ALDH1A1TDP1TSHRCYP3A4ALOX15
SCHEMBL29561089 0.80 TSHR (0.51) ALDH1A1TDP1TSHRCYP3A4ALOX15
SCHEMBL17688824 0.79 ALDH1A1 (0.46) ALDH1A1TDP1TSHRCYP3A4ALOX15
SCHEMBL2084778 0.79 ALDH1A1 (0.48) ALDH1A1TDP1TSHRCYP3A4ALOX15
SCHEMBL1644833 0.79 ALDH1A1 (0.47) ALDH1A1TDP1TSHRCYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-20130317057-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME LLC 2013-11-28 US disclosed
EP-2595482-A1 ALDOSTERONE SYNTHASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-29 EP disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130317057-A1 ALDOSTERONE SYNTHASE INHIBITORS HSD11B1, CYP11B2, HSD11B2 ALDH1A1 300/4885TDP1 3119/4885TSHR 2880/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.