Oxymesterone

Oxymesterone

SCHEMBL4317992

CC1(O)CC[C@H]2[C@@H]3CCC4=C(O)C(=O)CC[C@]4(C)[C@@H]3CC[C@@]21C

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.69
TSHR P16473 1/20 0.69
THPO P40225 1/20 0.69
HIF1A Q16665 1/20 0.69
TDP1 Q9NUW8 1/20 0.69
SHBG P04278 3/20 0.60
ALDH1A1 P00352 1/20 0.60
NR3C1 P04150 1/20 0.60
PGR P06401 1/20 0.60
ADRA1A P35348 1/20 0.60
HTR2B P41595 1/20 0.60
CYP19A1 P11511 12/20 0.53
LMNA P02545 1/20 0.49
MAPT P10636 1/20 0.49
POLB P06746 1/20 0.48
MAPK1 P28482 1/20 0.48
SRD5A1 P18405 1/20 0.46
SRD5A2 P31213 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxymesterone SCHEMBL4317989 1.00 CYP3A4 (0.69) CYP3A4TSHRTHPOHIF1ATDP1
Oxymesterone SCHEMBL141603 1.00 CYP3A4 (0.69) CYP3A4TSHRTHPOHIF1ATDP1
SCHEMBL9542851 0.90 SHBG (0.57) CYP3A4TSHRTHPOHIF1ATDP1
SCHEMBL9542854 0.90 SHBG (0.57) CYP3A4TSHRTHPOHIF1ATDP1
SCHEMBL9542574 0.88 CYP3A4 (0.67) CYP3A4TSHRTHPOHIF1ATDP1
SCHEMBL9542566 0.88 CYP3A4 (0.67) CYP3A4TSHRTHPOHIF1ATDP1
SCHEMBL23801605 0.87 SHBG (0.57) CYP3A4TSHRTHPOHIF1ATDP1
SCHEMBL9544690 0.87 SHBG (0.57) CYP3A4TSHRTHPOHIF1ATDP1
SCHEMBL7951228 0.87 SHBG (0.57) CYP3A4TSHRTHPOHIF1ATDP1
SCHEMBL9542783 0.87 CYP19A1 (0.68) CYP3A4TSHRTHPOHIF1ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150152348-A1 SYSTEMS AND METHODS FOR COLLECTING, TRANSPORTING AND REPURPOSING OR DESTROYING UNUSED PHARMACEUTICALS SHARPS COMPLIANCE, INC. OF TEXAS 2015-06-04 US disclosed
US-20090123571-A1 Method of treating men with testosterone supplement and 5alpha-reductase inhibitor MERCK SHARP & DOHME CORP. 2009-05-14 US disclosed
EP-1865955-A4 METHOD OF TREATING MEN WITH TESTOSTERONE SUPPLEMENT AND 5ALPHA-REDUCTASE INHIBITOR MERCK & CO INC (US) 2009-04-15 EP disclosed
US-20080207601-A1 Methods of and Compositions For the Prevention of Anxiety, Substance Abuse, and Dependence HYTHIAM , INC. (US) 2008-08-28 US disclosed
EP-1868593-A2 IMPROVED METHODS OF AND COMPOSITIONS FOR THE PREVENTION OF ANXIETY, SUBSTANCE ABUSE, AND DEPENDENCE Hythiam, Inc. (US) 2007-12-26 EP disclosed
EP-1865955-A2 METHOD OF TREATING MEN WITH TESTOSTERONE SUPPLEMENT AND 5ALPHA-REDUCTASE INHIBITOR Merck & Co., Inc. (US) 2007-12-19 EP disclosed
WO-2006110642-A2 IMPROVED METHODS OF AND COMPOSITIONS FOR THE PREVENTION OF ANXIETY, SUBSTANCE ABUSE, AND DEPENDENCE HYTHIAM, INC. (US) 2006-10-19 WO disclosed
WO-2006104762-A2 METHOD OF TREATING MEN WITH TESTOSTERONE SUPPLEMENT AND 5ALPHA-REDUCTASE INHIBITOR MERCK & CO., INC. (US) 2006-10-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090123571-A1 Method of treating men with testosterone supplement and 5alpha-reductase inhibitor ADRA1D, ADRB1, AGER CYP3A4 1077/4885TSHR 629/4885THPO 2926/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.