SCHEMBL4319700

SCHEMBL4319700

O=C(O)c1ccc(C=Cc2ccccn2)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.48
KDM6B O15054 1/20 0.48
KDM4A O75164 1/20 0.48
KDM5C P41229 1/20 0.48
KDM4C Q9H3R0 1/20 0.48
KDM2A Q9Y2K7 1/20 0.48
KDM3A Q9Y4C1 1/20 0.48
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ATM Q13315 1/20 0.46
NTRK3 Q16288 2/20 0.44
HTR2A P28223 2/20 0.42
KCNH2 Q12809 2/20 0.42
HTR2C P28335 1/20 0.42
NTRK1 P04629 1/20 0.42
NTRK2 Q16620 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4319695 1.00 KDM4E (0.48) KDM4EKDM6BKDM4AKDM5CKDM4C
SCHEMBL4316427 0.84 ALOX15 (0.52) KDM4ENPC1RAB9AMEN1KMT2A
SCHEMBL4316421 0.84 ALOX15 (0.52) KDM4ENPC1RAB9AMEN1KMT2A
SCHEMBL22553033 0.80 NFE2L2 (0.55) RAB9AHTR2AKCNH2HTR2CSRD5A2
SCHEMBL709588 0.75 MEN1 (0.55) KDM4ENPC1RAB9AMEN1KMT2A
SCHEMBL709589 0.75 MEN1 (0.55) KDM4ENPC1RAB9AMEN1KMT2A
SCHEMBL6264887 0.75 TTR (0.58) KDM4EKDM6BKDM4AKDM5CKDM4C
SCHEMBL22887384 0.75 TTR (0.58) KDM4EKDM6BKDM4AKDM5CKDM4C
SCHEMBL4714352 0.74 NFE2L2 (0.64) KDM4ENPC1RAB9AMEN1KMT2A
SCHEMBL4714353 0.74 NFE2L2 (0.64) KDM4ENPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566781-B2 Imidazopyridine compound BANYU PHARMACEUTICAL CO., LTD. (JP) 2009-07-28 US disclosed
US-20070249659-A1 melanin concentrating hormone receptor antagonist; preventing or treating vascular system diseases, nervous system disorders, metabolic disorders, urogenital diseases, respiratory diseases disorders; N-(2-ethyl-3-methylimidazo[1,2-a]pyridin-6-yl)-3-fluoro-4-(pyridin-2-ylmethoxy)benzamide BANYU PHARMACEUTICAL., LTD. (JP) 2007-10-25 US disclosed
EP-1748048-A1 IMIDAZOPYRIDINE COMPOUND BANYU PHARMACEUTICAL CO., LTD. (JP) 2007-01-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070249659-A1 melanin concentrating hormone receptor antagonist; preventing or treating vascular system diseases, nervous system disorders, metabolic disorders, urogenital diseases, respiratory diseases disorders; N-(2-ethyl-3-methylimidazo[1,2-a]pyridin-6-yl)-3-fluoro-4-(pyridin-2-ylmethoxy)benzamide MC1R, MCHR2, MCHR1 KDM4E 1794/4885KDM6B 2344/4885KDM4A 1528/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.