SCHEMBL4324539

SCHEMBL4324539

COC(=O)c1ccc2c(-c3ccccc3)cn(CCOCC(=O)O)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.44
CNR1 P21554 2/20 0.41
CNR2 P34972 2/20 0.41
EGFR P00533 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
TSHR P16473 1/20 0.41
F2RL3 Q96RI0 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GLA P06280 1/20 0.40
HPGD P15428 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
PTGS2 P35354 1/20 0.40
CA12 O43570 4/20 0.40
CA1 P00915 4/20 0.40
CA2 P00918 4/20 0.40
CA9 Q16790 4/20 0.40
CPT2 P23786 1/20 0.40
CPT1A P50416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4331800 0.88 SCN9A (0.40) SCN9ACNR1CNR2EGFRL3MBTL1
SCHEMBL13578024 0.86 CPT2 (0.47) MEN1KMT2AALDH1A1CPT2CPT1A
SCHEMBL13577917 0.85 RXFP1 (0.42) SCN9ACNR1CNR2L3MBTL1F2RL3
SCHEMBL13578018 0.85 CPT2 (0.46) SCN9ATSHRF2RL3MEN1KMT2A
SCHEMBL13577941 0.84 ASH1L (0.48) SCN9ACNR2EGFRL3MBTL1F2RL3
SCHEMBL4326615 0.84 SCN9A (0.49) SCN9ACNR2EGFRL3MBTL1F2RL3
SCHEMBL4333426 0.84 ALDH1A1 (0.48) SCN9AEGFRL3MBTL1F2RL3MEN1
Hydrochloric Acid SCHEMBL4326712 0.84 ASH1L (0.47) SCN9ACNR2EGFRL3MBTL1F2RL3
SCHEMBL4324605 0.84 KDM4E (0.42) CNR1CNR2L3MBTL1TSHRKMT2A
SCHEMBL13577916 0.84 ALDH1A1 (0.48) MEN1KMT2AALDH1A1HPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009147121-A1 CARBOXYL SUBSTITUTED INDOLES FOR USE AS PPAR ALPHA MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-10 WO disclosed
WO-2009147121-A1 CARBOXYL SUBSTITUTED INDOLES FOR USE AS PPAR ALPHA MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-10 WO disclosed