SCHEMBL4332057

SCHEMBL4332057

CCCCc1cccc(COC(=O)Oc2ccccc2)c1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IAPP P10997 3/20 0.44
ALOX5 P09917 1/20 0.43
PTGS2 P35354 1/20 0.43
BID P55957 3/20 0.41
MCL1 Q07820 3/20 0.41
PPARA Q07869 3/20 0.41
BCL2L1 Q07817 2/20 0.41
BAK1 Q16611 2/20 0.41
KAT8 Q9H7Z6 2/20 0.41
PPARG P37231 2/20 0.41
EP300 Q09472 1/20 0.41
KAT2A Q92830 1/20 0.41
KAT2B Q92831 1/20 0.41
KAT5 Q92993 1/20 0.41
SAE1 Q9UBE0 1/20 0.41
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
PTGER1 P34995 1/20 0.38
PTGER4 P35408 1/20 0.38
PTGER3 P43115 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4342474 0.92 IAPP (0.41) IAPPALOX5PPARAPPARGGABRA1
SCHEMBL4343854 0.88 GABRA1 (0.52) IAPPPPARGGABRA1GABRB2
SCHEMBL1006616 0.87 IAPP (0.51) IAPPALOX5PTGS2BIDMCL1
SCHEMBL2165406 0.82 HMGB1 (0.51) ALOX5PTGS2BIDMCL1PPARA
SCHEMBL4335272 0.80 GABRA1 (0.54) GABRA1GABRB2
SCHEMBL6151612 0.80 MEN1 (0.42) ALOX5BCL2L1
SCHEMBL3178976 0.79 ALOX5 (0.39) IAPPALOX5PTGS2BIDMCL1
SCHEMBL2887703 0.78 IAPP (0.49) IAPPALOX5PTGS2GABRA1GABRB2
SCHEMBL9389206 0.78 CYP4F2 (0.47) IAPPBIDMCL1PPARABCL2L1
SCHEMBL16395117 0.78 THRA (0.47) BIDMCL1PPARABCL2L1BAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3247734-B1 PREPARATION OF HIGHLY HEAT-RESISTANT (EO)POIYCARBONATES BY THE TRANSESTERIFICATION METHOD COVESTRO INTELLECTUAL PROPERTY GMBH & CO KG (DE) 2022-08-31 EP disclosed
US-10370491-B2 Preparation of highly heat-resistant (co)polycarbonates by the transesterification method COVESTRO DEUTSCHLAND AG (DE) 2019-08-06 US disclosed
US-20170369642-A1 Preparation of Highly Heat-Resistant (Co)Polycarbonates by the Transesterification Method COVESTRO DEUTSCHLAND AG (DE) 2017-12-28 US disclosed
EP-3247734-A1 PREPARATION OF HIGHLY HEAT-RESISTANT (EO)POIYCARBONATES BY THE TRANSESTERIFICATION METHOD Covestro Deutschland AG (DE) 2017-11-29 EP disclosed
WO-2016116480-A1 PREPARATION OF HIGHLY HEAT-RESISTANT (EO)POIYCARBONATES BY THE TRANSESTERIFICATION METHOD COVESTRO DEUTSCHLAND AG (DE) 2016-07-28 WO disclosed
US-20090117314-A1 PROCESS FOR THE PREPARATION OF POLYCARBONATE BY THE MELT TRANSESTERIFICATION METHOD BAYER MATERIALSCIENCE AG (DE) 2009-05-07 US disclosed
US-7259223-B2 Process for the production of polycarbonate GENERAL ELECTRIC COMPANY (US) 2007-08-21 US disclosed
EP-1360220-B1 PROCESS FOR THE PRODUCTION OF POLYCARBONATE GEN ELECTRIC (US) 2007-01-31 EP disclosed
US-20040220352-A1 Process for the production of polycarbonate SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2004-11-04 US disclosed
EP-1360220-A2 PROCESS FOR THE PRODUCTION OF POLYCARBONATE GENERAL ELECTRIC COMPANY (US) 2003-11-12 EP disclosed
US-20020132957-A1 Process for the production of polycarbonate GENERAL ELECTRIC COMPANY 2002-09-19 US disclosed
WO-2002060855-A2 PROCESS FOR THE PRODUCTION OF POLYCARBONATE GENERAL ELECTRIC COMPANY (US) 2002-08-08 WO disclosed