SCHEMBL433503

SCHEMBL433503

Fc1ccc(-c2c(F)[c]ccc2Cl)c(F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.34
HTR5A P47898 2/20 0.33
IDO1 P14902 2/20 0.33
AGXT P21549 2/20 0.33
MAPK13 O15264 3/20 0.32
MAPK12 P53778 3/20 0.32
MAPK11 Q15759 3/20 0.32
ALDH1A1 P00352 2/20 0.31
NISCH Q9Y2I1 1/20 0.31
ALOX15 P16050 1/20 0.31
CNR1 P21554 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
USP2 O75604 1/20 0.30
DHFR P00374 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
LMNA P02545 1/20 0.30
TTR P02766 1/20 0.30
ALB P02768 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8704011 0.88 NISCH (0.38) MAPK14NISCHKDM4EGRM2
SCHEMBL435281 0.86 KMO (0.34) GRM2
SCHEMBL432706 0.84 IDO1 (0.35) MAPK14IDO1AGXTALDH1A1KDM4E
SCHEMBL17514735 0.80
SCHEMBL17514551 0.79 NISCH (0.37) MAPK14NISCHGRM2
SCHEMBL434140 0.79 CYP1A2 (0.34) IDO1ALDH1A1KDM4E
SCHEMBL432660 0.77 ALDH1A1 (0.34) MAPK14HTR5AIDO1AGXTMAPK13
SCHEMBL1304581 0.77 IDO1 (0.33) MAPK14IDO1AGXTMAPK13MAPK12
SCHEMBL435101 0.77 AHR (0.40) ALDH1A1KDM4EHSD17B10
SCHEMBL17514836 0.74 NISCH (0.38) MAPK14NISCHKDM4EGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed