SCHEMBL435281

SCHEMBL435281

Fc1[c]ccc(Cl)c1-c1ccc(Cl)cc1F

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.34
HSD11B1 P28845 2/20 0.34
EGLN2 Q96KS0 1/20 0.33
GRM2 Q14416 2/20 0.33
PTGS2 P35354 1/20 0.33
AHR P35869 1/20 0.32
S100A4 P26447 1/20 0.31
PDE4A P27815 2/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL433574 0.88 KMO (0.35) KMOHSD11B1EGLN2GRM2PTGS2
SCHEMBL435101 0.88 AHR (0.40) HSD11B1AHRTP53
SCHEMBL433503 0.86 MAPK14 (0.34) GRM2
SCHEMBL17514805 0.86 GRM2 (0.35) KMOHSD11B1EGLN2GRM2PTGS2
SCHEMBL435121 0.79 AHR (0.39) HSD11B1AHRTP53
SCHEMBL434140 0.79 CYP1A2 (0.34) HSD11B1
SCHEMBL8704011 0.77 NISCH (0.38) HSD11B1GRM2HTR2AHTR2CHTR2B
SCHEMBL17514822 0.77 KMO (0.35) KMOHSD11B1EGLN2GRM2AHR
SCHEMBL17514854 0.77 GRM2 (0.38) KMOHSD11B1EGLN2GRM2S100A4
SCHEMBL433543 0.77 PTGS2 (0.36) KMOHSD11B1EGLN2GRM2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016026830-A1 NOVEL FUNGICIDAL PYRAZOLE DERIVATIVES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-02-25 WO disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed