SCHEMBL433557

SCHEMBL433557

Fc1cc(Cl)ccc1[C]1CCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
KMO O15229 2/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
EGLN2 Q96KS0 1/20 0.37
PDE4A P27815 2/20 0.36
PDE4B Q07343 2/20 0.36
PDE4C Q08493 2/20 0.36
PDE4D Q08499 1/20 0.36
GRM2 Q14416 2/20 0.36
S100A4 P26447 1/20 0.35
HTT P42858 1/20 0.35
HSD11B1 P28845 1/20 0.35
FASN P49327 1/20 0.34
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
CYP19A1 P11511 1/20 0.33
ACP1 P24666 1/20 0.33
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL434241 0.98 KMT2A (0.43) KMT2AKMOHTR2AHTR2CHTR2B
SCHEMBL434517 0.96 KMO (0.38) KMT2AKMOHTR2AHTR2CHTR2B
SCHEMBL433272 0.91 KMO (0.40) KMT2AKMOHTR2AHTR2CHTR2B
SCHEMBL23638850 0.79 S100A4 (0.46) KMOEGLN2GRM2S100A4HSD11B1
SCHEMBL30598347 0.79 S100A4 (0.46) KMOEGLN2GRM2S100A4HSD11B1
SCHEMBL436723 0.78 MAOA (0.41) KMT2AKMOPDE4BPDE4DCYP11B1
SCHEMBL432638 0.78 AHR (0.48) S100A4HTTHSD11B1
SCHEMBL434607 0.77 AHR (0.47) HSD11B1
SCHEMBL435253 0.77 MAOA (0.42) KMT2APDE4BPDE4DHTTCYP11B1
SCHEMBL435076 0.74 ALDH1A1 (0.39) KMT2AKMOCYP11B1CYP11B2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016026830-A1 NOVEL FUNGICIDAL PYRAZOLE DERIVATIVES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-02-25 WO disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed