SCHEMBL433687

SCHEMBL433687

O=C(NC(CN1CCCC1)c1ccccc1)C1(c2ccc3ccc(=O)[nH]c3c2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.40
ROCK2 O75116 3/20 0.39
ROCK1 Q13464 3/20 0.39
GPR88 Q9GZN0 1/20 0.37
RAB9A P51151 2/20 0.36
MITF O75030 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36
GFER P55789 1/20 0.36
PAX8 Q06710 1/20 0.36
ATM Q13315 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
AURKA O14965 3/20 0.36
AURKB Q96GD4 2/20 0.36
CDC7 O00311 1/20 0.36
CHEK1 O14757 1/20 0.36
JAK2 O60674 1/20 0.36
PAK4 O96013 1/20 0.36
NTRK1 P04629 1/20 0.36
PRKCB P05771 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15385522 1.00 TRPV1 (0.40) TRPV1ROCK2ROCK1GPR88RAB9A
SCHEMBL459835 0.94 ROCK2 (0.39) TRPV1ROCK2ROCK1GPR88RAB9A
SCHEMBL459836 0.94 ROCK2 (0.39) TRPV1ROCK2ROCK1GPR88RAB9A
SCHEMBL459306 0.88 ROCK2 (0.40) ROCK2ROCK1GPR88RAB9AMITF
SCHEMBL10083028 0.88 ROCK2 (0.40) ROCK2ROCK1GPR88RAB9AMITF
SCHEMBL434875 0.86 TRPV1 (0.42) TRPV1ROCK2ROCK1GPR88RAB9A
SCHEMBL15385515 0.86 TRPV1 (0.42) TRPV1ROCK2ROCK1GPR88RAB9A
SCHEMBL435831 0.83 HSD11B1 (0.50) GPR88RAB9AMITFALDH1A1HTT
SCHEMBL15385492 0.83 HSD11B1 (0.50) GPR88RAB9AMITFALDH1A1HTT
SCHEMBL461061 0.82 ROCK2 (0.53) TRPV1ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed