SCHEMBL459306

SCHEMBL459306

O=C(NC(CN1CCCC1)c1ccccc1)C1(c2ccc3[nH]c(=O)[nH]c3c2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.40
ROCK1 Q13464 2/20 0.40
AURKA O14965 3/20 0.38
AURKB Q96GD4 2/20 0.38
CDC7 O00311 1/20 0.38
CHEK1 O14757 1/20 0.38
JAK2 O60674 1/20 0.38
PAK4 O96013 1/20 0.38
NTRK1 P04629 1/20 0.38
PRKCB P05771 1/20 0.38
INSR P06213 1/20 0.38
RET P07949 1/20 0.38
KIT P10721 1/20 0.38
FGFR1 P11362 1/20 0.38
PRKACA P17612 1/20 0.38
FLT4 P35916 1/20 0.38
KDR P35968 1/20 0.38
JAK3 P52333 1/20 0.38
PDK1 Q15118 1/20 0.38
STK26 Q9P289 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10083028 1.00 ROCK2 (0.40) ROCK2ROCK1AURKAAURKBCDC7
SCHEMBL433687 0.88 TRPV1 (0.40) ROCK2ROCK1AURKAAURKBCDC7
SCHEMBL15385522 0.88 TRPV1 (0.40) ROCK2ROCK1AURKAAURKBCDC7
SCHEMBL459835 0.87 ROCK2 (0.39) ROCK2ROCK1AURKAAURKBCDC7
SCHEMBL459836 0.87 ROCK2 (0.39) ROCK2ROCK1AURKAAURKBCDC7
SCHEMBL434875 0.86 TRPV1 (0.42) ROCK2ROCK1AURKAAURKBCDC7
SCHEMBL15385515 0.86 TRPV1 (0.42) ROCK2ROCK1AURKAAURKBCDC7
SCHEMBL435831 0.83 HSD11B1 (0.50) GPR88MAPK1MITFALDH1A1HTT
SCHEMBL15385492 0.83 HSD11B1 (0.50) GPR88MAPK1MITFALDH1A1HTT
SCHEMBL433254 0.82 MAPK1 (0.42) ROCK2ROCK1AURKAAURKBCDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012410-A2 KAPPA OPIOID RECEPTOR AGONISTS DR. REDDY'S LABORATORIES LTD. (IN) 2012-01-26 WO disclosed