Bromodiolone

Bromodiolone

SCHEMBL433993

O=c1oc2ccccc2c(O)c1C(CC(O)c1ccc(-c2ccc(Br)cc2)cc1)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 1.00
CYP2C9 P11712 7/20 0.64
VKORC1 Q9BQB6 3/20 0.64
NQO1 P15559 3/20 0.60
CTSK P43235 1/20 0.58
KDM4E B2RXH2 2/20 0.55
HSD17B10 Q99714 2/20 0.55
ALDH1A1 P00352 1/20 0.55
ALB P02768 1/20 0.55
PCSK7 Q16549 1/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
POLB P06746 1/20 0.54
CYP3A4 P08684 1/20 0.54
TOP1 P11387 1/20 0.53
TOP2A P11388 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromodiolone SCHEMBL29362860 1.00 THRB (1.00) THRBCYP2C9VKORC1NQO1CTSK
SCHEMBL18962174 0.89 THRB (0.80) THRBCYP2C9VKORC1NQO1KDM4E
SCHEMBL18802989 0.89 THRB (0.80) THRBCYP2C9VKORC1NQO1KDM4E
SCHEMBL8335244 0.88 THRB (0.78) THRBCYP2C9VKORC1NQO1CTSK
SCHEMBL5933914 0.86 THRB (0.75) THRBCYP2C9VKORC1NQO1CTSK
SCHEMBL8337124 0.85 CYP2C9 (0.77) THRBCYP2C9VKORC1NQO1CTSK
SCHEMBL8334663 0.84 THRB (0.72) THRBCYP2C9VKORC1NQO1CTSK
SCHEMBL8332272 0.83 THRB (0.71) THRBCYP2C9VKORC1NQO1CTSK
SCHEMBL8333320 0.82 THRB (0.70) THRBCYP2C9VKORC1NQO1CTSK
SCHEMBL8523615 0.82 THRB (0.70) THRBCYP2C9VKORC1NQO1CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4428 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137082-A1 FUNGICIDAL COMPOSITIONS COMPRISING FLUDIOXONIL SYNGENTA CROP PROTECTION AG (CH) 2026-05-21 US claimed
EP-2991482-B1 PACKAGED RODENTICIDAL BAIT BASF AGRO BV (NL) 2026-05-20 EP claimed
EP-3175865-B1 FUNCTIONAL PARTICLES, PROCESS TO OBTAIN THEM, AND THEIR APPLICATIONS SMART INOVATION LDA (PT) 2026-04-15 EP claimed
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
EP-3578543-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-08-20 EP claimed
EP-3578541-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY, AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-05-28 EP claimed
US-12279613-B2 Attractant blend compositions, devices and methods for attracting female mice VARNER ELANA (US) 2025-04-22 US claimed
CN-119667065-A Kit and method for screening 74 toxic drugs in blood 华中科技大学同济医学院附属同济医院 2025-03-21 CN claimed
CN-119586629-A Preparation method of fluorescent rodenticide 安徽康宇生物科技工程有限公司 2025-03-11 CN claimed
US-5720951-A GROUND CEREAL BASE; WATER-SOLUBLE FILM-FORMING BINDER; AGGLOMERATED GRANULES ZENECA LIMITED (GB) 1998-02-24 US claimed
CN-1170503-A Raticide WANG YINGSHAN (CN) 1998-01-21 CN claimed
EP-0772391-A1 A RODENTICIDE BAIT ZENECA LIMITED (GB) 1997-05-14 EP claimed
WO-1996003037-A1 A RODENTICIDE BAIT ZENECA LIMITED (GB) 1996-02-08 WO claimed
EP-0594653-A1 RODENT BAIT PACKAGE ZENECA LIMITED (GB) 1994-05-04 EP claimed
WO-1993001712-A1 RODENT BAIT PACKAGE ZENECA LIMITED (GB) 1993-02-04 WO claimed
EP-0475551-A2 Bait block LIPHATECH, INC. (US) 1992-03-18 EP claimed
EP-0088051-B1 RODENTICIDAL BAIT CIBA-GEIGY AG (CH) 1986-11-12 EP claimed
US-4310536-A Rodenticidal compositions LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1982-01-12 US claimed
US-3980634-A Phthalimidyl-azo aniline type compounds and polyester fibers dyed therewith EASTMAN KODAK COMPANY (US) 1976-09-14 US claimed