SCHEMBL4347491

SCHEMBL4347491

CC(=O)c1cc(NCc2ccccc2Sc2ccc3cccnc3c2)cc(Cl)c1O

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSD P07339 8/20 0.40
HDAC6 Q9UBN7 1/20 0.36
KDR P35968 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
NOTUM Q6P988 1/20 0.33
GAA P10253 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
ALOX12 P18054 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33
NPC1 O15118 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6230126 0.94 CTSD (0.44) CTSDHDAC6NOTUMTRPV1EGLN1
SCHEMBL4347648 0.90 GAA (0.38) CTSDHDAC6SMN1; SMN2L3MBTL1GAA
SCHEMBL6230128 0.88 CTSD (0.39) CTSDHDAC6KDRNOTUMALOX12
SCHEMBL6230133 0.86 CTSD (0.37) CTSDHDAC6KDRNOTUMTRPV1
SCHEMBL4350092 0.86 CTSD (0.38) CTSDHDAC6KDRSMN1; SMN2L3MBTL1
SCHEMBL6223808 0.85 CTSD (0.39) CTSDHDAC6KDRNOTUMNPC1
SCHEMBL4349874 0.84 GAA (0.33) CTSDHDAC6SMN1; SMN2L3MBTL1GAA
SCHEMBL4348911 0.84 MEN1 (0.39) CTSDSMN1; SMN2L3MBTL1MEN1KMT2A
SCHEMBL6227080 0.84 GAA (0.36) CTSDHDAC6SMN1; SMN2L3MBTL1GAA
SCHEMBL4346923 0.83 SLC6A4 (0.43) CTSDHDAC6SMN1; SMN2GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed