SCHEMBL4343702

SCHEMBL4343702

CC(C)(C)N(S)C(=O)Nc1cc(Cl)c(O)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.43
APEX1 P27695 1/20 0.41
NPC1 O15118 2/20 0.40
MAPT P10636 2/20 0.40
MCL1 Q07820 1/20 0.40
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
P2RX5 Q93086 1/20 0.38
P2RX4 Q99571 1/20 0.38
P2RX7 Q99572 1/20 0.38
P2RX2 Q9UBL9 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
POLB P06746 1/20 0.37
GAA P10253 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
TTR P02766 2/20 0.35
TSHR P16473 1/20 0.34
HTT P42858 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4349894 0.86 GAA (0.40) DHODHAPEX1NPC1MAPTMCL1
SCHEMBL4347099 0.83 APEX1 (0.49) APEX1MAPTALDH1A1MEN1KMT2A
SCHEMBL13737975 0.83 APEX1 (0.64) APEX1NPC1MAPTALDH1A1KDM4E
SCHEMBL4353361 0.82 XDH (0.39) ALDH1A1P2RX7GAATDP1HTT
SCHEMBL6566879 0.81 DHODH (0.43) DHODHAPEX1NPC1MAPTMCL1
SCHEMBL4343499 0.81 ALDH1A1 (0.39) MAPTALDH1A1KDM4EHPGDMEN1
SCHEMBL4344516 0.80 HSPA5 (0.48) NPC1MAPTMCL1ALDH1A1KDM4E
SCHEMBL10883879 0.78 APEX1 (0.66) DHODHAPEX1NPC1MAPTMCL1
SCHEMBL4350112 0.75 LMNA (0.33) MAPTKMT2APOLBGAATSHR
SCHEMBL9402610 0.74 GAA (0.59) DHODHNPC1MAPTMCL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed