SCHEMBL4353361

SCHEMBL4353361

CC(C)(C)N(S)C(=O)Nc1cc(F)c(O)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.39
SLC22A12 Q96S37 1/20 0.39
GAA P10253 2/20 0.38
ALDH1A1 P00352 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
P2RX1 P51575 1/20 0.33
P2RX7 Q99572 1/20 0.33
TP53 P04637 1/20 0.33
AR P10275 1/20 0.32
HTT P42858 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347727 0.84 HTT (0.38) TP53ARHTT
SCHEMBL4343499 0.82 ALDH1A1 (0.39) GAAALDH1A1TDP1HTT
SCHEMBL4343702 0.82 DHODH (0.43) GAAALDH1A1TDP1P2RX7HTT
SCHEMBL4358260 0.77 HTT (0.34) GAAALDH1A1HTT
SCHEMBL22200943 0.75 GAA (0.59) XDHSLC22A12GAAALDH1A1TDP1
SCHEMBL4346777 0.75 HTT (0.38) GAAALDH1A1TP53HTT
SCHEMBL4346269 0.75 CXCR2 (0.39) ALDH1A1P2RX1P2RX7HTT
SCHEMBL4349894 0.73 GAA (0.40) GAAALDH1A1TDP1P2RX7HTT
SCHEMBL4351163 0.72 HTT (0.58) XDHSLC22A12GAAALDH1A1TDP1
SCHEMBL7751129 0.72 LMNA (0.59) XDHSLC22A12GAAALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed