SCHEMBL4346971

SCHEMBL4346971

O=[N+]([O-])c1cc(NC(=S)Nc2ccc(Cl)cc2)ccc1O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPIA P62937 1/20 0.58
P2RX1 P51575 1/20 0.54
MEN1 O00255 6/20 0.53
KMT2A Q03164 6/20 0.53
MAPT P10636 8/20 0.51
ALDH1A1 P00352 6/20 0.51
HTT P42858 4/20 0.51
GAA P10253 4/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
HPGD P15428 2/20 0.51
NPSR1 Q6W5P4 2/20 0.48
LMNA P02545 4/20 0.48
ALOX12 P18054 2/20 0.48
HSP90AA1 P07900 1/20 0.48
XBP1 P17861 1/20 0.48
EGFR P00533 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
AURKB Q96GD4 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4344002 0.90 PPIA (0.56) PPIAP2RX1MEN1KMT2AMAPT
SCHEMBL4353650 0.87 MAPT (0.63) PPIAMEN1KMT2AMAPTALDH1A1
SCHEMBL4356349 0.87 MEN1 (0.62) P2RX1MEN1KMT2AMAPTHTT
SCHEMBL4345484 0.82 HRAS (0.54) PPIAMEN1KMT2AMAPTALDH1A1
SCHEMBL4345759 0.80 ALDH1A1 (0.51) PPIAMEN1KMT2AMAPTALDH1A1
SCHEMBL28529066 0.79 MAPK1 (0.53) PPIAP2RX1MEN1KMT2AMAPT
SCHEMBL4357526 0.79 ALDH1A1 (0.50) PPIAMEN1KMT2AMAPTALDH1A1
SCHEMBL25348807 0.78 P2RX1 (0.85) P2RX1MEN1KMT2AMAPTALDH1A1
SCHEMBL4342020 0.77 MAPT (0.57) P2RX1MEN1KMT2AMAPTHTT
SCHEMBL25249421 0.77 MAPT (0.68) P2RX1MEN1KMT2AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed