SCHEMBL434428

SCHEMBL434428

C[C](C)Cc1ccc(Cl)cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.41
ERCC4 Q92889 1/20 0.41
HTR2A P28223 4/20 0.39
TP53 P04637 1/20 0.39
HTR1A P08908 1/20 0.39
HTR7 P34969 1/20 0.39
HTR6 P50406 1/20 0.39
CXCR3 P49682 1/20 0.37
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 2/20 0.37
POLB P06746 1/20 0.37
TSHR P16473 1/20 0.37
SLC6A4 P31645 5/20 0.36
KCNH2 Q12809 4/20 0.36
IDO1 P14902 2/20 0.36
SLC6A2 P23975 2/20 0.36
CYP3A4 P08684 2/20 0.36
MEN1 O00255 1/20 0.36
SLC22A1 O15245 1/20 0.36
USP2 O75604 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13187181 0.85 ERCC1 (0.39) ERCC1ERCC4HTR2ATP53HTR1A
SCHEMBL19030836 0.85 ERCC1 (0.46) ERCC1ERCC4HTR2ATP53HTR1A
SCHEMBL9730240 0.82 ERCC1 (0.40) ERCC1ERCC4HTR2ATP53HTR1A
SCHEMBL435206 0.79 IDO1 (0.54) ERCC1ERCC4ALDH1A1IDO1CYP3A4
SCHEMBL434355 0.79 IDO1 (0.48) ALDH1A1IDO1SMN1; SMN2P2RX7
SCHEMBL29434734 0.78 KEAP1 (0.50) ERCC1ERCC4HTR2ATP53HTR1A
SCHEMBL348979 0.78 KEAP1 (0.50) ERCC1ERCC4HTR2ATP53HTR1A
SCHEMBL1488965 0.78 ERCC1 (0.47) ERCC1ERCC4HTR2ATP53HTR1A
SCHEMBL9921231 0.78 KCNH2 (0.45) HTR2ATP53HTR1AHTR7HTR6
SCHEMBL5266985 0.77 ICMT (0.46) ERCC1ERCC4HTR2ATP53HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016026830-A1 NOVEL FUNGICIDAL PYRAZOLE DERIVATIVES BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2016-02-25 WO disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed