SCHEMBL4346828

SCHEMBL4346828

Cc1ccccc1NC(=O)Nc1ccc(O)c(F)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDX3X O00571 3/20 0.66
RAB9A P51151 10/20 0.58
KMT2A Q03164 6/20 0.58
MAPT P10636 5/20 0.58
MEN1 O00255 5/20 0.58
HTT P42858 3/20 0.58
NPC1 O15118 9/20 0.58
NFKB1 P19838 1/20 0.58
NFKB2 Q00653 1/20 0.58
RELA Q04206 1/20 0.58
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
ALDH1A1 P00352 1/20 0.54
IMPDH2 P12268 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.52
STING1 Q86WV6 1/20 0.52
KCNJ6 P48051 1/20 0.51
KCNJ5 P48544 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4354644 0.85 DDX3X (0.65) DDX3XRAB9AKMT2AMAPTMEN1
SCHEMBL5071986 0.84 RAB9A (0.71) DDX3XRAB9AKMT2AMAPTMEN1
SCHEMBL4353772 0.84 KMT2A (0.56) DDX3XRAB9AKMT2AMAPTMEN1
SCHEMBL4360021 0.83 DDX3X (0.66) DDX3XRAB9AKMT2AMAPTMEN1
SCHEMBL4351601 0.82 MAOA (0.59) RAB9AKMT2AMAPTMEN1HTT
SCHEMBL4356409 0.81 MAPT (0.62) RAB9AKMT2AMAPTMEN1HTT
SCHEMBL11918074 0.80 DDX3X (1.00) DDX3XRAB9AKMT2AMAPTMEN1
SCHEMBL1659299 0.80 DDX3X (1.00) DDX3XRAB9AKMT2AMAPTMEN1
SCHEMBL4354193 0.79 DDX3X (0.65) DDX3XRAB9AKMT2AMAPTMEN1
SCHEMBL4341716 0.79 RAB9A (0.62) RAB9AKMT2AMEN1NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed