SCHEMBL4353993

SCHEMBL4353993

O=C(NCc1ccc(C(F)(F)F)cc1)Nc1cc(Cl)c(O)c(Cl)c1

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTOR P42345 5/20 0.67
NAMPT P43490 2/20 0.60
PRMT3 O60678 1/20 0.54
CNR1 P21554 1/20 0.53
RORC P51449 3/20 0.53
TRPV1 Q8NER1 1/20 0.52
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA7 P43166 1/20 0.51
CA9 Q16790 1/20 0.51
RAB9A P51151 2/20 0.49
POLB P06746 1/20 0.49
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347012 0.88 MTOR (0.56) MTORNAMPTPRMT3CNR1RORC
SCHEMBL4348431 0.87 MTOR (0.68) MTORNAMPTPRMT3CNR1RORC
SCHEMBL4348348 0.85 MTOR (0.69) MTORNAMPTPRMT3CNR1RORC
SCHEMBL6229028 0.85 MTOR (0.56) MTORNAMPTPRMT3CNR1RORC
SCHEMBL4357497 0.84 MEN1 (0.61) MAPT
SCHEMBL4350068 0.84 MTOR (0.67) MTORNAMPTPRMT3CNR1TRPV1
SCHEMBL4350084 0.84 MTOR (0.56) MTORNAMPTPRMT3CNR1TRPV1
SCHEMBL4348880 0.83 EPHX2 (0.69) MTORTRPV1CA1CA2CA9
SCHEMBL4350061 0.82 MTOR (0.55) MTORCA1CA2CA9RAB9A
SCHEMBL4357504 0.80 TRPV1 (0.61) MTORNAMPTTRPV1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed