SCHEMBL434762

SCHEMBL434762

O=C(Nc1cc(Cl)c(Cl)nc1OC1CNC1)c1ccnc(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 1/20 0.45
KCNH2 Q12809 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45
TAS1R3 Q7RTX0 2/20 0.42
TAS1R1 Q7RTX1 2/20 0.42
TAS1R2 Q8TE23 2/20 0.42
SUCNR1 Q9BXA5 1/20 0.40
GSK3B P49841 3/20 0.40
WNT1 P04628 2/20 0.40
DYRK1A Q13627 2/20 0.40
CLK2 P49760 1/20 0.40
CLK3 P49761 1/20 0.40
GSK3A P49840 1/20 0.39
BRAF P15056 1/20 0.38
MAPK14 Q16539 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL434415 0.88 SLC6A3 (0.45) SLC6A3KCNH2TAAR1TAS1R3TAS1R1
SCHEMBL434455 0.86 SLC6A3 (0.45) SLC6A3KCNH2TAAR1TAS1R3TAS1R1
SCHEMBL431125 0.86 SLC6A3 (0.45) SLC6A3KCNH2TAAR1TAS1R3TAS1R1
SCHEMBL433524 0.84 RAF1 (0.43) SLC6A3KCNH2TAAR1BRAF
SCHEMBL432002 0.80 TAS1R3 (0.38) TAS1R3TAS1R1TAS1R2GSK3BGSK3A
SCHEMBL1727518 0.77 SLC6A3 (0.45) SLC6A3KCNH2TAAR1TAS1R3TAS1R1
SCHEMBL432744 0.77 KDM4E (0.39) SLC6A3KCNH2TAAR1
SCHEMBL432151 0.74 KDM4E (0.37) SLC6A3KCNH2TAAR1
SCHEMBL431263 0.72 HDAC1 (0.37) TAS1R3TAS1R1TAS1R2GSK3BGSK3A
SCHEMBL433484 0.72 HDAC1 (0.37) TAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012366-A1 PESTICIDAL 3-(ARYLOXY)AZACYCLOALKANES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-01-26 WO disclosed