SCHEMBL4347648

SCHEMBL4347648

Oc1c(Cl)cc(NCc2ccccc2Sc2ccc3cccnc3c2)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.38
HDAC6 Q9UBN7 1/20 0.37
KDM4E B2RXH2 5/20 0.37
ALDH1A1 P00352 4/20 0.37
NPC1 O15118 3/20 0.37
LMNA P02545 3/20 0.37
GFER P55789 2/20 0.37
HPGD P15428 2/20 0.37
HTT P42858 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 6/20 0.36
KMT2A Q03164 6/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
NR4A2 P43354 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
ALOX12 P18054 2/20 0.36
CTSD P07339 1/20 0.35
MAPT P10636 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6227080 0.92 GAA (0.36) GAAHDAC6KDM4EALDH1A1NPC1
SCHEMBL4347491 0.90 CTSD (0.40) GAAHDAC6NPC1HTTRAB9A
SCHEMBL4349874 0.90 GAA (0.33) GAAHDAC6KDM4EALDH1A1NPC1
SCHEMBL4358574 0.90 HDAC6 (0.40) HDAC6KDM4EALDH1A1NPC1LMNA
SCHEMBL4357398 0.88 MEN1 (0.42) GAAHDAC6KDM4EALDH1A1NPC1
SCHEMBL4347748 0.88 LMNA (0.41) GAAHDAC6KDM4EALDH1A1NPC1
SCHEMBL6223808 0.87 CTSD (0.39) HDAC6ALDH1A1NPC1HTTRAB9A
SCHEMBL4347116 0.87 GAA (0.43) GAAKDM4EALDH1A1LMNAGFER
SCHEMBL4344502 0.87 MEN1 (0.43) GAAKDM4EALDH1A1HPGDHTT
SCHEMBL6230126 0.85 CTSD (0.44) HDAC6ALDH1A1NPC1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed