SCHEMBL6230126

SCHEMBL6230126

CC(=O)Nc1ccc(Sc2ccccc2CNc2cc(Cl)c(O)c(C(C)=O)c2)cc1.CC(=O)c1cc(NCc2ccccc2Sc2ccc3cccnc3c2)cc(Cl)c1O

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSD P07339 10/20 0.44
NPC1 O15118 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
MAPT P10636 2/20 0.34
EGLN1 Q9GZT9 1/20 0.34
NOTUM Q6P988 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
GRM4 Q14833 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347491 0.94 CTSD (0.40) CTSDNPC1HTTRAB9AHDAC6
SCHEMBL6230128 0.94 CTSD (0.39) CTSDNPC1HTTRAB9AHDAC6
SCHEMBL6223808 0.91 CTSD (0.39) CTSDNPC1HTTRAB9AHDAC6
SCHEMBL4351090 0.88 LMNA (0.41) CTSDHTTRAB9AMAPTALDH1A1
SCHEMBL6230133 0.87 CTSD (0.37) CTSDHDAC6NOTUMTRPV1
SCHEMBL4347648 0.85 GAA (0.38) CTSDNPC1HTTRAB9AHDAC6
SCHEMBL4346978 0.82 MAPT (0.41) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL4350092 0.81 CTSD (0.38) CTSDNPC1HTTRAB9AHDAC6
SCHEMBL4346923 0.80 SLC6A4 (0.43) CTSDHDAC6MAPTALDH1A1LMNA
SCHEMBL4343453 0.80 SMN1; SMN2 (0.43) RAB9AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed