SCHEMBL4349347

SCHEMBL4349347

COc1ccc(C[C@H](N)CN(C(=O)O)C(C)(C)C)cc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.53
SLC6A4 P31645 1/20 0.47
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
TDP1 Q9NUW8 1/20 0.41
EPHX1 P07099 1/20 0.41
TPH1 P17752 1/20 0.41
POLB P06746 1/20 0.41
ACHE P22303 1/20 0.41
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4349354 1.00 LDHA (0.53) LDHASLC6A4CYP1A2CYP2D6CYP2C19
SCHEMBL14860143 0.85 EPHX1 (0.48) EPHX1ALDH1A1HTT
SCHEMBL14860145 0.85 EPHX1 (0.48) EPHX1ALDH1A1HTT
SCHEMBL1527219 0.85 EPHX1 (0.48) EPHX1ALDH1A1HTT
SCHEMBL3777016 0.85 LDHA (0.52) LDHASLC6A4CYP1A2CYP2D6CYP2C19
SCHEMBL4343817 0.84 RIPK1 (0.40) TDP1EPHX1TPH1
SCHEMBL4343822 0.84 RIPK1 (0.40) TDP1EPHX1TPH1
SCHEMBL4359730 0.84 SLC6A4 (0.50) SLC6A4CYP1A2CYP2D6CYP2C19PPARG
SCHEMBL4359724 0.84 SLC6A4 (0.50) SLC6A4CYP1A2CYP2D6CYP2C19PPARG
SCHEMBL4347700 0.82 ANPEP (0.40) CYP1A2CYP2C19ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2070928-A1 7-azaindol-3-ylacrylamides active as kinase inhibitors NERVIANO MEDICAL SCIENCES S.r.l. (IT) 2009-06-17 EP disclosed